Generation of Fcabs targeting human and murine LAG-3 as building blocks for novel bispecific antibody therapeutics.


Journal

Methods (San Diego, Calif.)
ISSN: 1095-9130
Titre abrégé: Methods
Pays: United States
ID NLM: 9426302

Informations de publication

Date de publication:
01 02 2019
Historique:
received: 18 06 2018
revised: 31 08 2018
accepted: 04 09 2018
pubmed: 13 9 2018
medline: 28 11 2019
entrez: 13 9 2018
Statut: ppublish

Résumé

The immunoglobulin superfamily protein lymphocyte-activation gene 3 (LAG-3) participates in immune suppression and has been identified as a suitable target for cancer therapies. In order to generate bispecific antibodies targeting LAG-3, Fcabs (Fc-region with antigen binding) targeting human and murine LAG-3 were generated from phage libraries. These Fcabs bind to LAG-3, inhibiting its interaction with MHC class II, and induce IL-2 production in a T cell assay. Bispecific antibodies, known as mAb

Identifiants

pubmed: 30208333
pii: S1046-2023(18)30103-8
doi: 10.1016/j.ymeth.2018.09.003
pii:
doi:

Substances chimiques

Antibodies, Bispecific 0
Antigens, CD 0
Immunoglobulin Fc Fragments 0
Lymphocyte Activation Gene 3 Protein 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

60-69

Informations de copyright

Copyright © 2018 Elsevier Inc. All rights reserved.

Auteurs

Katy L Everett (KL)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom. Electronic address: katy.everett@f-star.com.

Matthew Kraman (M)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Francisca P G Wollerton (FPG)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Carlo Zimarino (C)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Katarzyna Kmiecik (K)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Miguel Gaspar (M)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Sarka Pechouckova (S)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Natalie L Allen (NL)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Jacqueline F Doody (JF)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

Mihriban Tuna (M)

F-star Biotechnology Ltd, Eddeva B920, Babraham Research Campus, Cambridge CB22 3AT, United Kingdom.

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Classifications MeSH