Endothelium-dependent and endothelium-independent vasorelaxant effects of tiliacorinine 12'-O-acetate and mechanisms on isolated rat aorta.
Endothelium-dependent
Endothelium-independent
Hypertension
Tiliacorinine 12′-O-acetate
Vasorelaxant effect
Journal
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie
ISSN: 1950-6007
Titre abrégé: Biomed Pharmacother
Pays: France
ID NLM: 8213295
Informations de publication
Date de publication:
Jan 2019
Jan 2019
Historique:
received:
19
06
2018
revised:
13
11
2018
accepted:
14
11
2018
entrez:
16
12
2018
pubmed:
16
12
2018
medline:
2
4
2019
Statut:
ppublish
Résumé
Tiliacorinine 12'-O-acetate is a modified analog of Tiliacorinine, a major compound in Tiliacora triandra. The present study explored the vasorelaxation property of tiliacorinine 12'-O-acetate and its mechanism in isolated rat aorta using the organ bath technique. Tiliacorinine 12'-O-acetate exhibited concentration-dependent (10
Identifiants
pubmed: 30551466
pii: S0753-3322(18)34141-6
doi: 10.1016/j.biopha.2018.11.062
pii:
doi:
Substances chimiques
Benzylisoquinolines
0
Vasodilator Agents
0
tiliacorinine
0
Acetic Acid
Q40Q9N063P
Types de publication
Comparative Study
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Pagination
2090-2099Informations de copyright
Copyright © 2018 The Authors. Published by Elsevier Masson SAS.. All rights reserved.