Fluoromethylene Transfer from Diarylfluoromethylsulfonium Salts: Synthesis of Fluorinated Epoxides.

Johnson-Corey-Chaykovsky reaction fluorinated epoxides fluoromethylenation fluorooxiranes sulfur fluoromethylylide

Journal

Chemistry (Weinheim an der Bergstrasse, Germany)
ISSN: 1521-3765
Titre abrégé: Chemistry
Pays: Germany
ID NLM: 9513783

Informations de publication

Date de publication:
12 Mar 2019
Historique:
received: 22 01 2019
pubmed: 27 1 2019
medline: 27 1 2019
entrez: 26 1 2019
Statut: ppublish

Résumé

Diarylfluoromethyl sulfonium salts are efficient fluoromethylene transfer reagents equivalent to fluorocarbene, which is difficult to access. This was demonstrated by the development of a monofluorinated Johnson-Corey-Chaykovsky reaction with ketones and aldehydes, delivering uncommon 2-unsubstituted fluoroepoxides. This is the first evidence for the feasibility of sulfur fluoromethylylide and its action as a reaction intermediate.

Identifiants

pubmed: 30681208
doi: 10.1002/chem.201900349
doi:

Types de publication

Journal Article

Langues

eng

Pagination

3786-3789

Subventions

Organisme : European Regional Development Fund
ID : Nr.1.1.1.5/17/A/003

Informations de copyright

© 2019 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim.

Auteurs

Janis Veliks (J)

Latvian Institute of Organic Synthesis, Aizkraukles 21, LV-1006, Riga, Latvia.

Armands Kazia (A)

Latvian Institute of Organic Synthesis, Aizkraukles 21, LV-1006, Riga, Latvia.

Classifications MeSH