The Use of a Microfluidic Device to Encapsulate a Poorly Water-Soluble Drug CoQ


Journal

Journal of pharmaceutical sciences
ISSN: 1520-6017
Titre abrégé: J Pharm Sci
Pays: United States
ID NLM: 2985195R

Informations de publication

Date de publication:
08 2019
Historique:
received: 06 03 2019
revised: 01 04 2019
accepted: 02 04 2019
pubmed: 9 4 2019
medline: 18 8 2020
entrez: 9 4 2019
Statut: ppublish

Résumé

A number of drugs that are currently on the market, as well as new candidates for drugs, are poorly water soluble. Because of this, a need exists to develop drug formulations that will permit the expanded use of such drugs. The use of liposomes and lipid nanoparticles for drug delivery has attracted attention as a technique for solubilizing molecules that are poorly water soluble, but this technique faces serious scale-up risks. In this study, we report on attempts to encapsulate Coenzyme Q

Identifiants

pubmed: 30959057
pii: S0022-3549(19)30214-X
doi: 10.1016/j.xphs.2019.04.001
pii:
doi:

Substances chimiques

Lipids 0
Liposomes 0
Vitamins 0
Water 059QF0KO0R
Ubiquinone 1339-63-5
coenzyme Q10 EJ27X76M46

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

2668-2676

Informations de copyright

Copyright © 2019. Published by Elsevier Inc.

Auteurs

Mitsue Hibino (M)

Faculty of Pharmaceutical Sciences, Hokkaido University, 1-1 Kita-12, Nishi-6, Kita-ku, Sapporo 060-0812, Japan.

Yuma Yamada (Y)

Faculty of Pharmaceutical Sciences, Hokkaido University, 1-1 Kita-12, Nishi-6, Kita-ku, Sapporo 060-0812, Japan.

Naoki Fujishita (N)

Faculty of Pharmaceutical Sciences, Hokkaido University, 1-1 Kita-12, Nishi-6, Kita-ku, Sapporo 060-0812, Japan.

Yusuke Sato (Y)

Faculty of Pharmaceutical Sciences, Hokkaido University, 1-1 Kita-12, Nishi-6, Kita-ku, Sapporo 060-0812, Japan.

Masatoshi Maeki (M)

Faculty of Engineering, Hokkaido University, Kita-13, Nishi-8, Kita-ku, Sapporo 060-8628, Japan.

Manabu Tokeshi (M)

Faculty of Engineering, Hokkaido University, Kita-13, Nishi-8, Kita-ku, Sapporo 060-8628, Japan.

Hideyoshi Harashima (H)

Faculty of Pharmaceutical Sciences, Hokkaido University, 1-1 Kita-12, Nishi-6, Kita-ku, Sapporo 060-0812, Japan. Electronic address: harasima@pharm.hokudai.ac.jp.

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Classifications MeSH