Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515.
Journal
ACS medicinal chemistry letters
ISSN: 1948-5875
Titre abrégé: ACS Med Chem Lett
Pays: United States
ID NLM: 101521073
Informations de publication
Date de publication:
11 Apr 2019
11 Apr 2019
Historique:
received:
22
11
2018
accepted:
13
03
2019
entrez:
19
4
2019
pubmed:
19
4
2019
medline:
19
4
2019
Statut:
epublish
Résumé
Poly(ADP-ribose) polymerase-1 (PARP-1) is an enzyme involved in signaling and repair of DNA single strand breaks. PARP-1 employs NAD
Identifiants
pubmed: 30996792
doi: 10.1021/acsmedchemlett.8b00569
pmc: PMC6466814
doi:
Types de publication
Journal Article
Langues
eng
Pagination
534-538Déclaration de conflit d'intérêts
The authors declare no competing financial interest.
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