Development, Validation of LC-MS/MS Method and Determination of Pharmacokinetic Parameters of the Stroke Neuroprotectant Neurounina-1 in Beagle Dog Plasma After Intravenous Administration.

LC-MS/MS Na+/Ca2+ exchanger (NCX) beagle dog plasma neurounina-1 pharmacokinetics

Journal

Frontiers in pharmacology
ISSN: 1663-9812
Titre abrégé: Front Pharmacol
Pays: Switzerland
ID NLM: 101548923

Informations de publication

Date de publication:
2019
Historique:
received: 23 07 2018
accepted: 04 04 2019
entrez: 11 5 2019
pubmed: 11 5 2019
medline: 11 5 2019
Statut: epublish

Résumé

Neurounina-1 [chemical name: 7-nitro-5-phenyl-1-(pyrrolidin-1-ylmethyl)-1H-benzo[e][1,4]diazepin-2(3H)-one] is a new compound provided with relevant neuroprotective effect during stroke and in neonatal hypoxia by increasing the Na

Identifiants

pubmed: 31073288
doi: 10.3389/fphar.2019.00432
pmc: PMC6497007
doi:

Types de publication

Journal Article

Langues

eng

Pagination

432

Références

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pubmed: 15472108
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pubmed: 15602012
Cell Calcium. 2008 May;43(5):482-91
pubmed: 17884163
J Neurosci. 2008 Jan 30;28(5):1179-84
pubmed: 18234895
Mol Pharmacol. 2013 Jan;83(1):142-56
pubmed: 23066092
J Cereb Blood Flow Metab. 2016 Oct;36(10):1790-1803
pubmed: 26661211
J Cereb Blood Flow Metab. 2017 Jul;37(7):2539-2554
pubmed: 27683449
Neuropharmacology. 2018 Jun;135:180-191
pubmed: 29551690

Auteurs

Beatrice Severino (B)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Angela Corvino (A)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Ferdinando Fiorino (F)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Francesco Frecentese (F)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Elisa Perissutti (E)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Giuseppe Caliendo (G)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Vincenzo Santagada (V)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Elisa Magli (E)

Department of Pharmacy, School of Medicine, University of Naples Federico II, Naples, Italy.

Pasquale Molinaro (P)

Department of Neuroscience, Reproductive and Odontostomatological Sciences, School of Medicine, University of Naples Federico II, Naples, Italy.

Giuseppe Pignataro (G)

Department of Neuroscience, Reproductive and Odontostomatological Sciences, School of Medicine, University of Naples Federico II, Naples, Italy.

Lucio Annunziato (L)

IRCCS SDN, Naples, Italy.

Natalícia J Antunes (NJ)

Department of Pharmacology, Faculty of Medical Sciences, State University of Campinas, Campinas, Brazil.

Julio Rojas-Moscoso (J)

Department of Pharmacology, Faculty of Medical Sciences, State University of Campinas, Campinas, Brazil.

Noedi L de Freitas (NL)

Department of Pharmacology, Faculty of Medical Sciences, State University of Campinas, Campinas, Brazil.

Gustavo D Mendes (GD)

Department of Pharmacology, Faculty of Medical Sciences, Metropolitan University of Santos, Santos, Brazil.
Department of Pharmacology, Faculty of Medicine, São Leopoldo Mandic, Campinas, Brazil.
Faculty of Medicine, University of Mogi das Cruzes, Mogi das Cruzes, Brazil.

Gilberto De Nucci (G)

Department of Pharmacology, Faculty of Medical Sciences, State University of Campinas, Campinas, Brazil.
Department of Pharmacology, Faculty of Medicine, São Leopoldo Mandic, Campinas, Brazil.
Department of Pharmacology, Faculty of Medical Sciences, University of São Paulo, São Paulo, Brazil.

Classifications MeSH