Diazepam Accelerates GABA
GABAAR
benzodiazepine
diazepam
gephyrin
inhibitory synapse
mass spectrometry
trafficking
Journal
Frontiers in cellular neuroscience
ISSN: 1662-5102
Titre abrégé: Front Cell Neurosci
Pays: Switzerland
ID NLM: 101477935
Informations de publication
Date de publication:
2019
2019
Historique:
received:
17
01
2019
accepted:
08
04
2019
entrez:
14
5
2019
pubmed:
14
5
2019
medline:
14
5
2019
Statut:
epublish
Résumé
Despite 50+ years of clinical use as anxiolytics, anti-convulsants, and sedative/hypnotic agents, the mechanisms underlying benzodiazepine (BZD) tolerance are poorly understood. BZDs potentiate the actions of gamma-aminobutyric acid (GABA), the primary inhibitory neurotransmitter in the adult brain, through positive allosteric modulation of γ2 subunit containing GABA type A receptors (GABA
Identifiants
pubmed: 31080408
doi: 10.3389/fncel.2019.00163
pmc: PMC6497791
doi:
Types de publication
Journal Article
Langues
eng
Pagination
163Subventions
Organisme : NIMH NIH HHS
ID : F31 MH117839
Pays : United States
Organisme : NIMH NIH HHS
ID : R01 MH114908
Pays : United States
Organisme : NIMH NIH HHS
ID : R56 MH114908
Pays : United States
Organisme : NIGMS NIH HHS
ID : T32 GM008424
Pays : United States
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