Multicomponent Ugi Reaction of Indole- N-carboxylic Acids: Expeditious Access to Indole Carboxamide Amino Amides.


Journal

Organic letters
ISSN: 1523-7052
Titre abrégé: Org Lett
Pays: United States
ID NLM: 100890393

Informations de publication

Date de publication:
05 07 2019
Historique:
pubmed: 30 6 2019
medline: 30 6 2019
entrez: 29 6 2019
Statut: ppublish

Résumé

A novel multicomponent Ugi-type reaction for the synthesis of indole carboxamide amino amides from aldehydes, amines, isocyanides, and indole- N-carboxylic acids, which were simply prepared from indoles and CO

Identifiants

pubmed: 31247803
doi: 10.1021/acs.orglett.9b01871
doi:

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

5269-5272

Auteurs

Linwei Zeng (L)

Institute of Drug Discovery and Design, College of Pharmaceutical Sciences , Zhejiang University , Hangzhou 310058 , China.

Hironao Sajiki (H)

Laboratory of Organic Chemistry , Gifu Pharmaceutical University , Gifu 501-1196 , Japan.

Sunliang Cui (S)

Institute of Drug Discovery and Design, College of Pharmaceutical Sciences , Zhejiang University , Hangzhou 310058 , China.

Classifications MeSH