Desensitization of cAMP Accumulation via Human β3-Adrenoceptors Expressed in Human Embryonic Kidney Cells by Full, Partial, and Biased Agonists.

biased agonism cAMP desensitization extracellular signal-related kinase partial agonism β3-adrenoceptor

Journal

Frontiers in pharmacology
ISSN: 1663-9812
Titre abrégé: Front Pharmacol
Pays: Switzerland
ID NLM: 101548923

Informations de publication

Date de publication:
2019
Historique:
received: 24 02 2019
accepted: 09 05 2019
entrez: 3 7 2019
pubmed: 3 7 2019
medline: 3 7 2019
Statut: epublish

Résumé

β

Identifiants

pubmed: 31263412
doi: 10.3389/fphar.2019.00596
pmc: PMC6590479
doi:

Types de publication

Journal Article

Langues

eng

Pagination

596

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Auteurs

Katerina Okeke (K)

Department of Pharmacology, Johannes Gutenberg University Mainz, Mainz, Germany.
Department of Urology, University of Thessaly, Larissa, Greece.

Martina B Michel-Reher (MB)

Department of Pharmacology, Johannes Gutenberg University Mainz, Mainz, Germany.

Stavros Gravas (S)

Department of Urology, University of Thessaly, Larissa, Greece.

Martin C Michel (MC)

Department of Pharmacology, Johannes Gutenberg University Mainz, Mainz, Germany.

Classifications MeSH