Mannosylation of LNP Results in Improved Potency for Self-Amplifying RNA (SAM) Vaccines.


Journal

ACS infectious diseases
ISSN: 2373-8227
Titre abrégé: ACS Infect Dis
Pays: United States
ID NLM: 101654580

Informations de publication

Date de publication:
13 09 2019
Historique:
pubmed: 11 7 2019
medline: 18 6 2020
entrez: 11 7 2019
Statut: ppublish

Résumé

Mannosylation of Lipid Nanoparticles (LNP) can potentially enhance uptake by Antigen Presenting Cells, which are highly abundant in dermal tissues, to improve the potency of Self Amplifying mRNA (SAM) vaccines in comparison to the established unmodified LNP delivery system. In the current studies, we evaluated mannosylated LNP (MLNP), which were obtained by incorporation of a stable Mannose-cholesterol amine conjugate, for the delivery of an influenza (hemagglutinin) encoded SAM vaccine in mice, by both intramuscular and intradermal routes of administration. SAM MLNP exhibited

Identifiants

pubmed: 31290323
doi: 10.1021/acsinfecdis.9b00084
doi:

Substances chimiques

Hemagglutinin Glycoproteins, Influenza Virus 0
Immunoglobulin G 0
Influenza Vaccines 0
RNA, Messenger 0
Cholesterol 97C5T2UQ7J
Mannose PHA4727WTP

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1546-1558

Auteurs

Roshan Goswami (R)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Despo Chatzikleanthous (D)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Gustavo Lou (G)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Fabiola Giusti (F)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Alessandra Bonci (A)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Marianna Taccone (M)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Michela Brazzoli (M)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Simona Gallorini (S)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Ilaria Ferlenghi (I)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Francesco Berti (F)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Derek T O'Hagan (DT)

GSK , 14200 Shady Grove Road , Rockville, Maryland 20850 , United States.

Carlo Pergola (C)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Barbara C Baudner (BC)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

Roberto Adamo (R)

GSK , Via Fiorentina 1 , 53100 Siena , Italy.

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Classifications MeSH