Novel antimycobacterial C-21 amide derivatives of the antibiotic fusidic acid: synthesis, pharmacological evaluation and rationalization of media-dependent activity using molecular docking studies in the binding site of human serum albumin.
Journal
MedChemComm
ISSN: 2040-2511
Titre abrégé: Medchemcomm
Pays: England
ID NLM: 101531525
Informations de publication
Date de publication:
01 Jun 2019
01 Jun 2019
Historique:
received:
14
03
2019
accepted:
11
04
2019
entrez:
16
7
2019
pubmed:
16
7
2019
medline:
16
7
2019
Statut:
epublish
Résumé
Fusidic acid is a natural product antibiotic used clinically, primarily against staphylococcal infections. It has also exhibited antimycobacterial activity against
Identifiants
pubmed: 31303994
doi: 10.1039/c9md00161a
pii: c9md00161a
pmc: PMC6596249
doi:
Types de publication
Journal Article
Langues
eng
Pagination
961-969Références
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