Biodistribution and radiation dosimetry of [
Dosimetry
PET
PSMA
Prostate cancer
Journal
EJNMMI research
ISSN: 2191-219X
Titre abrégé: EJNMMI Res
Pays: Germany
ID NLM: 101560946
Informations de publication
Date de publication:
25 Jul 2019
25 Jul 2019
Historique:
received:
26
04
2019
accepted:
17
07
2019
entrez:
27
7
2019
pubmed:
28
7
2019
medline:
28
7
2019
Statut:
epublish
Résumé
We investigated the whole-body distribution and the radiation dosimetry of [ Ten patients with prostate cancer and biochemical recurrence or radiologic evidence of metastatic diseases were examined with 329-384 MBq (mean 359 ± 17 MBq) [ Physiologic radiotracer accumulation was observed in the salivary and lacrimal glands, liver, spleen, and intestines, in a pattern resembling the distribution known from other PSMA-tracers with excretion via urinary and biliary pathways. The effective dose from [ The highest TBR of [
Identifiants
pubmed: 31346821
doi: 10.1186/s13550-019-0540-7
pii: 10.1186/s13550-019-0540-7
pmc: PMC6658635
doi:
Types de publication
Journal Article
Langues
eng
Pagination
66Références
Prostate. 1999 Apr 1;39(1):28-35
pubmed: 10221263
J Nucl Med. 2005 Jun;46(6):1023-7
pubmed: 15937315
Clin Cancer Res. 2008 May 15;14(10):3036-43
pubmed: 18483369
J Med Chem. 2009 Jan 22;52(2):347-57
pubmed: 19111054
J Med Chem. 2010 Feb 25;53(4):1732-40
pubmed: 20088512
Clin Cancer Res. 2011 Dec 15;17(24):7645-53
pubmed: 22042970
Eur J Nucl Med Mol Imaging. 2012 Jun;39(6):1085-6
pubmed: 22310854
Bioconjug Chem. 2012 Apr 18;23(4):688-97
pubmed: 22369515
Appl Radiat Isot. 2013 Jun;76:55-62
pubmed: 23063597
J Nucl Med. 2012 Dec;53(12):1883-91
pubmed: 23203246
Radiat Prot Dosimetry. 2014 Dec;162(3):299-305
pubmed: 24353030
Org Biomol Chem. 2014 Oct 28;12(40):8094-9
pubmed: 25190038
J Nucl Med. 2015 Jun;56(6):855-61
pubmed: 25883128
Mol Imaging Biol. 2015 Aug;17(4):565-74
pubmed: 25896814
Mol Imaging Biol. 2015 Aug;17(4):575-84
pubmed: 26013479
Eur J Nucl Med Mol Imaging. 2016 Jan;43(1):42-51
pubmed: 26318602
J Med Chem. 2016 Mar 10;59(5):1761-75
pubmed: 26878194
J Nucl Med. 2017 Mar;58(3):425-431
pubmed: 27789722
Eur J Nucl Med Mol Imaging. 2017 Apr;44(4):678-688
pubmed: 27889802
J Nucl Med. 2017 Jun;58(6):947-952
pubmed: 27908968
J Nucl Med. 2019 Jun;60(6):817-823
pubmed: 30389823
J Pharmacol Exp Ther. 1998 Aug;286(2):1020-5
pubmed: 9694964