Successful Strategies for Mitigation of a Preclinical Signal for Phototoxicity in a DGAT1 Inhibitor.
Journal
ACS medicinal chemistry letters
ISSN: 1948-5875
Titre abrégé: ACS Med Chem Lett
Pays: United States
ID NLM: 101521073
Informations de publication
Date de publication:
08 Aug 2019
08 Aug 2019
Historique:
received:
18
03
2019
accepted:
20
06
2019
entrez:
16
8
2019
pubmed:
16
8
2019
medline:
16
8
2019
Statut:
epublish
Résumé
Diacylglycerol
Identifiants
pubmed: 31413796
doi: 10.1021/acsmedchemlett.9b00117
pmc: PMC6691483
doi:
Types de publication
Journal Article
Langues
eng
Pagination
1128-1133Déclaration de conflit d'intérêts
The authors declare no competing financial interest.
Références
Nat Genet. 2000 May;25(1):87-90
pubmed: 10802663
J Clin Invest. 2002 Apr;109(8):1049-55
pubmed: 11956242
Drug Saf. 2002;25(5):345-72
pubmed: 12020173
J Org Chem. 2007 Sep 14;72(19):7455-8
pubmed: 17696402
J Phys Chem A. 2008 Feb 14;112(6):1245-50
pubmed: 18198851
Pharmacol Ther. 2008 Jun;118(3):295-302
pubmed: 18508126
J Lipid Res. 2008 Nov;49(11):2283-301
pubmed: 18757836
J Lipid Res. 2010 Jul;51(7):1770-80
pubmed: 20147738
Drug Saf. 2011 Oct 1;34(10):821-37
pubmed: 21879777
Biochim Biophys Acta. 2011 Dec;1811(12):1011-20
pubmed: 21924378
Aging (Albany NY). 2012 Jan;4(1):13-27
pubmed: 22291164
J Clin Invest. 2012 Dec;122(12):4680-4
pubmed: 23114594
J Med Chem. 2013 Dec 27;56(24):9820-5
pubmed: 23919406
Regul Toxicol Pharmacol. 2014 Feb;68(1):70-5
pubmed: 24269723
Toxicol Sci. 2014 May;139(1):245-56
pubmed: 24519524
ACS Med Chem Lett. 2012 Apr 04;3(5):411-5
pubmed: 24900485
Nat Rev Endocrinol. 2015 Jun;11(6):352-62
pubmed: 25732519
J Clin Pharmacol. 2015 Sep;55(9):1031-41
pubmed: 25854859
Lipids Health Dis. 2015 Feb 18;14:8
pubmed: 25889044
Chemistry. 2015 Nov 9;21(46):16673-8
pubmed: 26395034
Photochem Photobiol Sci. 2016 Sep 31;15(9):1155-1162
pubmed: 27471837
J Med Chem. 2017 Jun 8;60(11):4657-4664
pubmed: 28498655
Cell Metab. 2017 Aug 1;26(2):407-418.e3
pubmed: 28768178
J Lipid Res. 2019 Jun;60(6):1112-1120
pubmed: 30936184
Endocrinol Metab Clin North Am. 1998 Sep;27(3):551-67, viii
pubmed: 9785052
Proc Natl Acad Sci U S A. 1998 Oct 27;95(22):13018-23
pubmed: 9789033