Second-Generation Inhibitors of the Mitochondrial Permeability Transition Pore with Improved Plasma Stability.
Animals
Dose-Response Relationship, Drug
Drug Stability
HeLa Cells
High-Throughput Screening Assays
Humans
Isoxazoles
/ blood
Mitochondrial Membrane Transport Proteins
/ antagonists & inhibitors
Mitochondrial Permeability Transition Pore
Molecular Structure
Muscular Dystrophies
/ drug therapy
Phenols
/ blood
Structure-Activity Relationship
Tumor Cells, Cultured
Zebrafish
calcium
click chemistry
inhibitors
mitochondria
muscular dystrophy
permeability transition pore
Journal
ChemMedChem
ISSN: 1860-7187
Titre abrégé: ChemMedChem
Pays: Germany
ID NLM: 101259013
Informations de publication
Date de publication:
17 10 2019
17 10 2019
Historique:
received:
22
06
2019
pubmed:
20
8
2019
medline:
10
9
2020
entrez:
20
8
2019
Statut:
ppublish
Résumé
Excessive mitochondrial matrix Ca
Identifiants
pubmed: 31423734
doi: 10.1002/cmdc.201900376
doi:
Substances chimiques
Isoxazoles
0
Mitochondrial Membrane Transport Proteins
0
Mitochondrial Permeability Transition Pore
0
Phenols
0
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
1771-1782Subventions
Organisme : Fondation Leducq
ID : 16CVD04
Pays : International
Informations de copyright
© 2019 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim.
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