Cell-Free Expression of Sodium Channel Domains for Pharmacology Studies. Noncanonical Spider Toxin Binding Site in the Second Voltage-Sensing Domain of Human Na

NMR spectroscopy cell-free expression channelopathies combinatorial selective labeling gating modifier ligand-receptor interactions sodium channel

Journal

Frontiers in pharmacology
ISSN: 1663-9812
Titre abrégé: Front Pharmacol
Pays: Switzerland
ID NLM: 101548923

Informations de publication

Date de publication:
2019
Historique:
received: 25 04 2019
accepted: 26 07 2019
entrez: 27 9 2019
pubmed: 27 9 2019
medline: 27 9 2019
Statut: epublish

Résumé

Voltage-gated sodium (Na

Identifiants

pubmed: 31555136
doi: 10.3389/fphar.2019.00953
pmc: PMC6737007
doi:

Types de publication

Journal Article

Langues

eng

Pagination

953

Subventions

Organisme : Medical Research Council
ID : G0802158
Pays : United Kingdom
Organisme : Medical Research Council
ID : G0900613
Pays : United Kingdom
Organisme : Medical Research Council
ID : MR/M006948/1
Pays : United Kingdom
Organisme : Medical Research Council
ID : G0400136
Pays : United Kingdom
Organisme : Medical Research Council
ID : G0600368
Pays : United Kingdom
Organisme : Medical Research Council
ID : G0400627
Pays : United Kingdom
Organisme : Medical Research Council
ID : G116/147
Pays : United Kingdom
Organisme : Medical Research Council
ID : G0601440
Pays : United Kingdom
Organisme : Wellcome Trust
ID : 209807/Z/17/Z
Pays : United Kingdom
Organisme : Wellcome Trust
ID : 212285/Z/18/Z
Pays : United Kingdom
Organisme : Medical Research Council
ID : G9805989
Pays : United Kingdom

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Auteurs

Mikhail Yu Myshkin (MY)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.

Roope Männikkö (R)

MRC Centre for Neuromuscular Diseases, Department of Molecular Neuroscience, UCL Institute of Neurology, London, United Kingdom.

Olesya A Krumkacheva (OA)

International Tomography Center SB RAS, Novosibirsk, Russia.

Dmitrii S Kulbatskii (DS)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.

Anton O Chugunov (AO)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.
School of Biological and Medical Physics, Moscow Institute of Physics and Technology (State University), Dolgoprudny, Russia.
International Laboratory for Supercomputer Atomistic Modelling and Multi-scale Analysis, National Research University Higher School of Economics, Moscow, Russia.

Antonina A Berkut (AA)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.

Alexander S Paramonov (AS)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.

Mikhail A Shulepko (MA)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.

Matvey V Fedin (MV)

International Tomography Center SB RAS, Novosibirsk, Russia.

Michael G Hanna (MG)

MRC Centre for Neuromuscular Diseases, Department of Molecular Neuroscience, UCL Institute of Neurology, London, United Kingdom.

Dimitri M Kullmann (DM)

Department of Clinical and Experimental Epilepsy, UCL Institute of Neurology, London, United Kingdom.

Elena G Bagryanskaya (EG)

N.N.Voroztsov Novosibirsk Institute of Organic Chemistry SB RAS, Novosibirsk, Russia.

Alexander S Arseniev (AS)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.
School of Biological and Medical Physics, Moscow Institute of Physics and Technology (State University), Dolgoprudny, Russia.

Mikhail P Kirpichnikov (MP)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.
Faculty of Biology, Lomonosov Moscow State University, Moscow, Russia.

Ekaterina N Lyukmanova (EN)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.
School of Biological and Medical Physics, Moscow Institute of Physics and Technology (State University), Dolgoprudny, Russia.

Alexander A Vassilevski (AA)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.
School of Biological and Medical Physics, Moscow Institute of Physics and Technology (State University), Dolgoprudny, Russia.

Zakhar O Shenkarev (ZO)

Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia.
School of Biological and Medical Physics, Moscow Institute of Physics and Technology (State University), Dolgoprudny, Russia.

Classifications MeSH