Non-Nucleoside Agonists of the Adenosine Receptors: An Overview.

adenosine receptor agonists adenosine receptors drug discovery ligand–target interaction non-nucleoside agonists purinergic receptors pyridine derivatives pyrimidine derivatives

Journal

Pharmaceuticals (Basel, Switzerland)
ISSN: 1424-8247
Titre abrégé: Pharmaceuticals (Basel)
Pays: Switzerland
ID NLM: 101238453

Informations de publication

Date de publication:
08 Oct 2019
Historique:
received: 09 09 2019
revised: 03 10 2019
accepted: 05 10 2019
entrez: 11 10 2019
pubmed: 11 10 2019
medline: 11 10 2019
Statut: epublish

Résumé

Potent and selective adenosine receptor (AR) agonists are of pharmacological interest for the treatment of a wide range of diseases and conditions. Among these derivatives, nucleoside-based agonists represent the great majority of molecules developed and reported to date. However, the limited availability of compounds selective for a specific AR subtype (i.e., A

Identifiants

pubmed: 31597388
pii: ph12040150
doi: 10.3390/ph12040150
pmc: PMC6958362
pii:
doi:

Types de publication

Journal Article Review

Langues

eng

Subventions

Organisme : undefined <span style="color:gray;font-size:10px;">undefined</span>
ID : 2015E8EMCM_008
Organisme : Italian Ministry of Research
ID : 2015E8EMCM_008

Déclaration de conflit d'intérêts

The authors declare no conflict of interest.

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Auteurs

Diego Dal Ben (D)

School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino (MC), Italy. diego.dalben@unicam.it.

Catia Lambertucci (C)

School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino (MC), Italy. catia.lambertucci@unicam.it.

Michela Buccioni (M)

School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino (MC), Italy. michela.buccioni@unicam.it.

Aleix Martí Navia (A)

School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino (MC), Italy. aleix.martinavia@unicam.it.

Gabriella Marucci (G)

School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino (MC), Italy. gabriella.marucci@unicam.it.

Andrea Spinaci (A)

School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino (MC), Italy. andrea.spinaci@unicam.it.

Rosaria Volpini (R)

School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, 62032 Camerino (MC), Italy. rosaria.volpini@unicam.it.

Classifications MeSH