Development of Triazinone-Based Condensing Reagents for Amide Formation.
Journal
The Journal of organic chemistry
ISSN: 1520-6904
Titre abrégé: J Org Chem
Pays: United States
ID NLM: 2985193R
Informations de publication
Date de publication:
06 12 2019
06 12 2019
Historique:
pubmed:
9
11
2019
medline:
9
11
2019
entrez:
9
11
2019
Statut:
ppublish
Résumé
Novel triazinone-based condensing reagents have been developed. The palladium-catalyzed O-N allylic rearrangement of 2-(allyloxy)-4,6-dichloro-1,3,5-triazine and subsequent regioselective substitution using alcohols and an amine afforded chlorotriazinones, which can be readily converted using
Identifiants
pubmed: 31701748
doi: 10.1021/acs.joc.9b01261
doi:
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM