Increased Paracetamol Bioavailability after Sleeve Gastrectomy: A Crossover Pre- vs. Post-Operative Clinical Trial.
bariatric surgery
drug absorption
gastric emptying
glucuronidation
laparoscopic sleeve gastrectomy
paracetamol (acetaminophen)
Journal
Journal of clinical medicine
ISSN: 2077-0383
Titre abrégé: J Clin Med
Pays: Switzerland
ID NLM: 101606588
Informations de publication
Date de publication:
12 Nov 2019
12 Nov 2019
Historique:
received:
24
09
2019
revised:
03
11
2019
accepted:
08
11
2019
entrez:
16
11
2019
pubmed:
16
11
2019
medline:
16
11
2019
Statut:
epublish
Résumé
Oral drug bioavailability may be significantly altered after laparoscopic sleeve gastrectomy (LSG), the most popular bariatric procedure worldwide. Paracetamol (acetaminophen) is the post-bariatric analgesic/antipyretic drug of choice. In this work we studied and analyzed the LSG effects on systemic bioavailability and pharmacokinetics of paracetamol after oral administration of solid vs. liquid dosage form. A 4-armed, pharmacokinetic, crossover trial was performed in patients enrolled for LSG. Single paracetamol dose (500 mg), as caplet (
Identifiants
pubmed: 31726725
pii: jcm8111949
doi: 10.3390/jcm8111949
pmc: PMC6912358
pii:
doi:
Types de publication
Journal Article
Langues
eng
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