Cathepsin B Turning Bioluminescence "On" for Tumor Imaging.
Animals
Biomarkers, Tumor
/ antagonists & inhibitors
Breast Neoplasms
/ diagnostic imaging
Cathepsin B
/ antagonists & inhibitors
Cell Line, Tumor
Diagnostic Imaging
/ methods
Dipeptides
/ pharmacology
Female
Gene Expression
Heterografts
Humans
Luminescent Measurements
Lysosomes
/ drug effects
Mice
Mice, Inbred BALB C
Mice, Nude
Molecular Probes
/ chemical synthesis
Journal
Analytical chemistry
ISSN: 1520-6882
Titre abrégé: Anal Chem
Pays: United States
ID NLM: 0370536
Informations de publication
Date de publication:
03 12 2019
03 12 2019
Historique:
pubmed:
16
11
2019
medline:
21
10
2020
entrez:
16
11
2019
Statut:
ppublish
Résumé
Cathepsin B (CTSB) is a lysosomal protease, and several human cancers are reported highly expressing CTSB. Many optical methods have been developed for CTSB detection but not a bioluminescence (BL) probe. Herein, a CTSB-specific bioluminescence probe
Identifiants
pubmed: 31726822
doi: 10.1021/acs.analchem.9b04254
doi:
Substances chimiques
Biomarkers, Tumor
0
CA 074 methyl ester
0
Dipeptides
0
Molecular Probes
0
CTSB protein, human
EC 3.4.22.1
Cathepsin B
EC 3.4.22.1
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM