Novel Hit Compounds as Putative Antifungals: The Case of
Aspergillus fumigatus
MFC
MIC
antifungal activity
molecular docking
molecular dynamics simulations
pharmacophore model
virtual screening
Journal
Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009
Informations de publication
Date de publication:
25 Oct 2019
25 Oct 2019
Historique:
received:
31
08
2019
revised:
19
10
2019
accepted:
23
10
2019
entrez:
17
11
2019
pubmed:
17
11
2019
medline:
24
4
2020
Statut:
epublish
Résumé
The prevalence of invasive fungal infections has been dramatically increased as the size of the immunocompromised population worldwide has grown.
Identifiants
pubmed: 31731542
pii: molecules24213853
doi: 10.3390/molecules24213853
pmc: PMC6864791
pii:
doi:
Substances chimiques
Antifungal Agents
0
Azoles
0
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : Ministry of Education, Science and Technological Development of Republic of Serbia
ID : 173032
Références
Microbiol Mol Biol Rev. 2011 Jun;75(2):213-67
pubmed: 21646428
Emerg Infect Dis. 2009 Jul;15(7):1068-76
pubmed: 19624922
Chem Pharm Bull (Tokyo). 2014;62(1):16-24
pubmed: 24390489
Chem Biol Drug Des. 2006 Jan;67(1):83-4
pubmed: 16492153
J Chem Inf Model. 2005 Jan-Feb;45(1):160-9
pubmed: 15667141
Drugs Today (Barc). 2015 Dec;51(12):705-18
pubmed: 26798851
Drugs. 2011 Dec 24;71(18):2405-19
pubmed: 22141384
Curr Opin Microbiol. 2018 Oct;45:70-76
pubmed: 29547801
J Fungi (Basel). 2016 Jun 06;2(2):null
pubmed: 29376934
N Engl J Med. 2002 Aug 8;347(6):408-15
pubmed: 12167683
J Med Chem. 2004 Mar 25;47(7):1739-49
pubmed: 15027865
Mayo Clin Proc. 2011 Aug;86(8):805-17
pubmed: 21803962
Biochem Pharmacol. 2017 Jun 1;133:86-96
pubmed: 27884742
Clin Infect Dis. 2010 Jun 15;50(12):1559-67
pubmed: 20450350
Mycoses. 2008 Sep;51 Suppl 4:2-15
pubmed: 18783559
Adv Drug Deliv Rev. 2001 Mar 1;46(1-3):3-26
pubmed: 11259830
J Mol Biol. 2010 Apr 9;397(4):1067-78
pubmed: 20149798
Curr Treat Options Infect Dis. 2014 Sep;6(3):309-325
pubmed: 25328449
J Chem Inf Model. 2005 Jan-Feb;45(1):177-82
pubmed: 15667143
Eur Respir Rev. 2011 Sep 1;20(121):156-74
pubmed: 21881144
Nat Rev Drug Discov. 2017 Sep;16(9):603-616
pubmed: 28496146
Proc Natl Acad Sci U S A. 2001 Mar 13;98(6):3068-73
pubmed: 11248033
Int J Antimicrob Agents. 2006 Nov;28(5):450-3
pubmed: 17034993
Biochim Biophys Acta. 2007 Mar;1770(3):467-77
pubmed: 16963187
Cold Spring Harb Perspect Med. 2014 Nov 10;5(7):a019752
pubmed: 25384768
J Clin Microbiol. 2001 Apr;39(4):1360-7
pubmed: 11283057
Molecules. 2015 Dec 19;20(12):22799-832
pubmed: 26703541
Microorganisms. 2017 Aug 22;5(3):null
pubmed: 28829379
Drug Discov Today. 2010 Jun;15(11-12):444-50
pubmed: 20362693
Antimicrob Agents Chemother. 2011 May;55(5):2483-6
pubmed: 21300838
J Chem Inf Model. 2010 Apr 26;50(4):572-84
pubmed: 20235588
Mycoses. 1998;41 Suppl 1:32-8
pubmed: 9717384
Clin Microbiol Rev. 1999 Apr;12(2):310-50
pubmed: 10194462
ChemMedChem. 2018 Feb 6;13(3):251-258
pubmed: 29235267
Trends Microbiol. 2003 Jun;11(6):272-9
pubmed: 12823944
Eur J Med Res. 2011 Apr 28;16(4):153-7
pubmed: 21486729
J Chem Inf Model. 2010 May 24;50(5):822-39
pubmed: 20423098
Antimicrob Agents Chemother. 2010 Oct;54(10):4225-34
pubmed: 20660663
J Med Chem. 2004 Mar 25;47(7):1750-9
pubmed: 15027866
J Comput Chem. 2012 Jan 15;33(2):119-33
pubmed: 21997754
Proteins. 2010 Jun;78(8):1950-8
pubmed: 20408171
Med Mycol. 2016 May;54(4):400-8
pubmed: 26768370