In Vitro Characterization and Stability Profiles of Antibody-Fluorophore Conjugates Derived from Interchain Cysteine Cross-Linking or Lysine Bioconjugation.

antibody–fluorophore conjugate bioconjugation fluorescence labelling

Journal

Pharmaceuticals (Basel, Switzerland)
ISSN: 1424-8247
Titre abrégé: Pharmaceuticals (Basel)
Pays: Switzerland
ID NLM: 101238453

Informations de publication

Date de publication:
02 Dec 2019
Historique:
received: 22 10 2019
revised: 22 11 2019
accepted: 25 11 2019
entrez: 8 12 2019
pubmed: 8 12 2019
medline: 8 12 2019
Statut: epublish

Résumé

Fluorescent labelling of monoclonal antibodies (mAbs) is classically performed by chemical bioconjugation methods. The most frequent labelling technique to generate antibody-fluorophore conjugates (AFCs) involves the bioconjugation onto the mAb lysines of a dye bearing an

Identifiants

pubmed: 31810248
pii: ph12040176
doi: 10.3390/ph12040176
pmc: PMC6958397
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Agence Nationale de la Recherche
ID : ANR-11-LABX-0029
Organisme : Agence Nationale de la Recherche
ID : ANR-10-LABX-53-01
Organisme : Région Centre Val de Loire
ID : -

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Auteurs

Camille Martin (C)

GICC EA7501, Equipe IMT, Université de Tours, UFR des Sciences Pharmaceutiques, 31 Avenue Monge, 37200 Tours, France.

Guillaume Brachet (G)

Laboratoire d'immunologie, CHRU Tours, 10 Bd Tonnelé, 37000 Tours, France.
GICC EA7501, Equipe FRAME, Université de Tours, 10 Bd Tonnelé, 37000 Tours, France.

Cyril Colas (C)

ICOA UMR 7311 CNRS, Université d'Orléans, Pôle de Chimie, Rue de Chartres, BP 6759, 45067 Orléans CEDEX 2, France.
CBM, UPR4301 CNRS, Rue Charles Sadron, 45071 Orléans, France.

Emilie Allard-Vannier (E)

NMNS EA 6295, 31 Avenue Monge, 37200 Tours, France.

Claire Kizlik-Masson (C)

GICC EA7501, Equipe FRAME, Université de Tours, 10 Bd Tonnelé, 37000 Tours, France.

Clara Esnault (C)

GICC EA7501, Equipe IMT, Université de Tours, UFR des Sciences Pharmaceutiques, 31 Avenue Monge, 37200 Tours, France.

Renaud Respaud (R)

INSERM U1100, Université de Tours, 10 Bd Tonnelé, 37000 Tours, France.

Caroline Denevault-Sabourin (C)

GICC EA7501, Equipe IMT, Université de Tours, UFR des Sciences Pharmaceutiques, 31 Avenue Monge, 37200 Tours, France.

Igor Chourpa (I)

NMNS EA 6295, 31 Avenue Monge, 37200 Tours, France.

Valérie Gouilleux-Gruart (V)

Laboratoire d'immunologie, CHRU Tours, 10 Bd Tonnelé, 37000 Tours, France.
GICC EA7501, Equipe FRAME, Université de Tours, 10 Bd Tonnelé, 37000 Tours, France.

Marie-Claude Viaud-Massuard (MC)

GICC EA7501, Equipe IMT, Université de Tours, UFR des Sciences Pharmaceutiques, 31 Avenue Monge, 37200 Tours, France.

Nicolas Joubert (N)

GICC EA7501, Equipe IMT, Université de Tours, UFR des Sciences Pharmaceutiques, 31 Avenue Monge, 37200 Tours, France.

Classifications MeSH