SerpinB3 Differently Up-Regulates Hypoxia Inducible Factors -1α and -2α in Hepatocellular Carcinoma: Mechanisms Revealing Novel Potential Therapeutic Targets.

HCC NEDD8 NEDDylation SerpinB3 hypoxia hypoxia inducible factors HIF-1α and HIF-2α

Journal

Cancers
ISSN: 2072-6694
Titre abrégé: Cancers (Basel)
Pays: Switzerland
ID NLM: 101526829

Informations de publication

Date de publication:
04 Dec 2019
Historique:
received: 04 11 2019
revised: 29 11 2019
accepted: 02 12 2019
entrez: 11 12 2019
pubmed: 11 12 2019
medline: 11 12 2019
Statut: epublish

Résumé

SerpinB3 (SB3) is a hypoxia and hypoxia-inducible factor (HIF)-2α-dependent cysteine-protease inhibitor up-regulated in hepatocellular carcinoma (HCC), released by cancer cells and able to stimulate proliferation and epithelial-to-mesenchymal-transition. Methods

Sections du résumé

BACKGROUND BACKGROUND
SerpinB3 (SB3) is a hypoxia and hypoxia-inducible factor (HIF)-2α-dependent cysteine-protease inhibitor up-regulated in hepatocellular carcinoma (HCC), released by cancer cells and able to stimulate proliferation and epithelial-to-mesenchymal-transition. Methods

Identifiants

pubmed: 31817100
pii: cancers11121933
doi: 10.3390/cancers11121933
pmc: PMC6966556
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Associazione Italiana per la Ricerca sul Cancro
ID : IG 2017 Id.20361
Organisme : EITB Maratoia
ID : BIO15/CA/014
Organisme : MIUR, Rome: 776 PRIN Project
ID : 2006067527
Organisme : University of Padova
ID : CPDA110795
Organisme : SAF2017-87301-R
ID : SAF2017-87301-R
Organisme : Gobierno 779 Vasco-Departamento de Salud
ID : 2013111114
Organisme : MINECO
ID : SEV-2016-0644

Déclaration de conflit d'intérêts

The authors declare no conflict of interest.

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Auteurs

Stefania Cannito (S)

Department of Clinical and Biological Sciences, Unit of Experimental Medicine & Clinical Pathology, University of Torino, 10125 Torino, Italy.

Beatrice Foglia (B)

Department of Clinical and Biological Sciences, Unit of Experimental Medicine & Clinical Pathology, University of Torino, 10125 Torino, Italy.

Gianmarco Villano (G)

Department of Surgery, Oncology and Gastroenterology, University of Padova, 35128 Padova, Italy.

Cristian Turato (C)

Veneto Institute of Oncology IOV-IRCCS, 35128 Padova, Italy.

Teresa C Delgado (TC)

Liver Disease and Metabolism Laboratory, CIC bioGUNE, Centro de Investigacion Biomedica en Red de Enfermedades Hepaticas y Digestivas (Ciberehd), Technology Park of Bizkaia, 48160 Derio, Bizkaia, Spain.

Elisabetta Morello (E)

Department of Clinical and Biological Sciences, Unit of Experimental Medicine & Clinical Pathology, University of Torino, 10125 Torino, Italy.

Fabrizio Pin (F)

Department of Clinical and Biological Sciences, Unit of Experimental Medicine & Clinical Pathology, University of Torino, 10125 Torino, Italy.

Erica Novo (E)

Department of Clinical and Biological Sciences, Unit of Experimental Medicine & Clinical Pathology, University of Torino, 10125 Torino, Italy.

Lucia Napione (L)

Department of Applied Science and Technology, Politecnico di Torino, 10129 Torino, Italy.
Laboratory of Vascular Oncology, Candiolo Cancer Institute-IRCCS, 10060 Candiolo, Italy.

Santina Quarta (S)

Department of Medicine, University of Padova, 35128 Padova, Italy.

Mariagrazia Ruvoletto (M)

Department of Surgery, Oncology and Gastroenterology, University of Padova, 35128 Padova, Italy.

Silvano Fasolato (S)

Department of Surgery, Oncology and Gastroenterology, University of Padova, 35128 Padova, Italy.

Giacomo Zanus (G)

Hepatobiliary Surgery, University of Padova, 35128 Padova, Italy.

Sebastiano Colombatto (S)

Department of Oncology, University of Torino, 10125 Torino, Italy.

Fernando Lopitz-Otsoa (F)

Liver Disease and Metabolism Laboratory, CIC bioGUNE, Centro de Investigacion Biomedica en Red de Enfermedades Hepaticas y Digestivas (Ciberehd), Technology Park of Bizkaia, 48160 Derio, Bizkaia, Spain.

David Fernández-Ramos (D)

Liver Disease and Metabolism Laboratory, CIC bioGUNE, Centro de Investigacion Biomedica en Red de Enfermedades Hepaticas y Digestivas (Ciberehd), Technology Park of Bizkaia, 48160 Derio, Bizkaia, Spain.

Federico Bussolino (F)

Laboratory of Vascular Oncology, Candiolo Cancer Institute-IRCCS, 10060 Candiolo, Italy.
Department of Oncology, University of Torino, 10125 Torino, Italy.

Salvatore Sutti (S)

Department of Health Sciences and Interdisciplinary Research Center for Autoimmune Diseases, University Amedeo Avogadro of East Piedmont, 28100 Novara, Italy.

Emanuele Albano (E)

Department of Health Sciences and Interdisciplinary Research Center for Autoimmune Diseases, University Amedeo Avogadro of East Piedmont, 28100 Novara, Italy.

Maria Luz Martínez-Chantar (ML)

Liver Disease and Metabolism Laboratory, CIC bioGUNE, Centro de Investigacion Biomedica en Red de Enfermedades Hepaticas y Digestivas (Ciberehd), Technology Park of Bizkaia, 48160 Derio, Bizkaia, Spain.

Patrizia Pontisso (P)

Department of Medicine, University of Padova, 35128 Padova, Italy.

Maurizio Parola (M)

Department of Clinical and Biological Sciences, Unit of Experimental Medicine & Clinical Pathology, University of Torino, 10125 Torino, Italy.

Classifications MeSH