Radioiodinated Nitroxide Derivative for the Detection of Lipid Radicals.


Journal

ACS medicinal chemistry letters
ISSN: 1948-5875
Titre abrégé: ACS Med Chem Lett
Pays: United States
ID NLM: 101521073

Informations de publication

Date de publication:
09 Jan 2020
Historique:
received: 09 09 2019
accepted: 03 12 2019
entrez: 16 1 2020
pubmed: 16 1 2020
medline: 16 1 2020
Statut: epublish

Résumé

Thus far, no accurate measurement technology has been developed to detect lipid alkyl radicals (lipid radicals), which cause lipid peroxidation. Therefore, we aimed to develop a nuclear medical imaging probe that can be taken up in the lipophilic site in cells such as biological membranes, by reacting specifically with the lipid radicals generated there. We designed and synthesized 4-(4-[

Identifiants

pubmed: 31938462
doi: 10.1021/acsmedchemlett.9b00416
pmc: PMC6956360
doi:

Types de publication

Journal Article

Langues

eng

Pagination

45-48

Informations de copyright

Copyright © 2019 American Chemical Society.

Déclaration de conflit d'intérêts

The authors declare no competing financial interest.

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Auteurs

Toshihide Yamasaki (T)

Laboratory of Biophysical Chemistry, Kobe Pharmaceutical University, 4-19-1 Motoyama-kita, Higashinada, Kobe 658-8558, Japan.

Risa Azuma (R)

Laboratory of Biophysical Chemistry, Kobe Pharmaceutical University, 4-19-1 Motoyama-kita, Higashinada, Kobe 658-8558, Japan.

Kohei Sano (K)

Laboratory of Biophysical Chemistry, Kobe Pharmaceutical University, 4-19-1 Motoyama-kita, Higashinada, Kobe 658-8558, Japan.

Masayuki Munekane (M)

Laboratory of Biophysical Chemistry, Kobe Pharmaceutical University, 4-19-1 Motoyama-kita, Higashinada, Kobe 658-8558, Japan.

Yuta Matsuoka (Y)

Physical Chemistry for Life Science Laboratory, Faculty of Pharmaceutical Sciences, Kyushu University, 3-1-1 Maidashi, Higashi-ku, Fukuoka 812-8582, Japan.

Ken-Ichi Yamada (KI)

Physical Chemistry for Life Science Laboratory, Faculty of Pharmaceutical Sciences, Kyushu University, 3-1-1 Maidashi, Higashi-ku, Fukuoka 812-8582, Japan.
AMED-CREST, Japan Agency for Medical Research and Development, Tokyo 100-0004, Japan.

Takahiro Mukai (T)

Laboratory of Biophysical Chemistry, Kobe Pharmaceutical University, 4-19-1 Motoyama-kita, Higashinada, Kobe 658-8558, Japan.

Classifications MeSH