Cabozantinib inhibits AXL- and MET-dependent cancer cell migration induced by growth-arrest-specific 6 and hepatocyte growth factor.

AXL receptor tyrosine kinase Cabozantinib Cancer cell migration Growth arrest-specific 6 Hepatocyte growth factor MET proto-oncogene-encoded receptor tyrosine kinase

Journal

Biochemistry and biophysics reports
ISSN: 2405-5808
Titre abrégé: Biochem Biophys Rep
Pays: Netherlands
ID NLM: 101660999

Informations de publication

Date de publication:
Mar 2020
Historique:
received: 26 09 2019
revised: 20 12 2019
accepted: 07 01 2020
entrez: 15 2 2020
pubmed: 15 2 2020
medline: 15 2 2020
Statut: epublish

Résumé

Cabozantinib is known as an inhibitor of receptor tyrosine kinases mainly targeting AXL receptor tyrosine kinase (AXL),

Identifiants

pubmed: 32055714
doi: 10.1016/j.bbrep.2020.100726
pii: S2405-5808(19)30267-5
pii: 100726
pmc: PMC7005370
doi:

Types de publication

Journal Article

Langues

eng

Pagination

100726

Commentaires et corrections

Type : ErratumIn

Informations de copyright

© 2020 The Authors.

Déclaration de conflit d'intérêts

T.H., A.K., T.M, MM, K.N and J.S. are employed by Takeda; H.T. is employed by Axcelead.

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Auteurs

Takahito Hara (T)

Innovation Promotion, Shonan Research Central Office, Research, Takeda Pharmaceutical Company Limited, 2-26-1 Muraoka-Higashi, Fujisawa-shi, Kanagawa, 251-8555, Japan.

Akiko Kimura (A)

Oncology Therapeutic Area Unit for Japan & Asia, Takeda Pharmaceutical Company Limited, 4-1-1 Dosho-machi Chuo-ku Osaka-shi, Osaka, 540-8645, Japan.

Tohru Miyazaki (T)

Department of Japan Medical Affairs, Japan Oncology Business Unit, Takeda Pharmaceutical Company Limited, 2-1-1 Nihonbashi-Honcho, Chuo-ku, Tokyo, 103-8668, Japan.

Hiroshi Tanaka (H)

Axcelead Drug Discovery Partners, Inc., 2-26-1Muraoka-Higashi, Fujisawa-shi, Kanagawa, 251-0012, Japan.

Megumi Morimoto (M)

Innovation Promotion, Shonan Research Central Office, Research, Takeda Pharmaceutical Company Limited, 2-26-1 Muraoka-Higashi, Fujisawa-shi, Kanagawa, 251-8555, Japan.

Katsuhiko Nakai (K)

Oncology Therapeutic Area Unit for Japan & Asia, Takeda Pharmaceutical Company Limited, 4-1-1 Dosho-machi Chuo-ku Osaka-shi, Osaka, 540-8645, Japan.

Junpei Soeda (J)

Department of Japan Medical Affairs, Japan Oncology Business Unit, Takeda Pharmaceutical Company Limited, 2-1-1 Nihonbashi-Honcho, Chuo-ku, Tokyo, 103-8668, Japan.

Classifications MeSH