Synthesis of Small-Molecule Fluorescent Probes for the In Vitro Imaging of Calcium-Activated Potassium Channel K

A549 Cells Binding Sites Boron Compounds / chemistry Cycloaddition Reaction Fluorescent Dyes / chemical synthesis Humans Intermediate-Conductance Calcium-Activated Potassium Channels / chemistry Ligands Microscopy, Fluorescence Molecular Dynamics Simulation
KCa3.1 channels cycloaddition fluorescent probes molecular modelling non-small cell lung cancer

Journal

Angewandte Chemie (International ed. in English)
ISSN: 1521-3773
Titre abrégé: Angew Chem Int Ed Engl
Pays: Germany
ID NLM: 0370543

Informations de publication

Date de publication:
18 05 2020
Historique:
received: 22 01 2020
revised: 19 02 2020
pubmed: 26 2 2020
medline: 12 3 2021
entrez: 26 2 2020
Statut: ppublish

Résumé

Small-molecule probes for the in vitro imaging of K

Identifiants

DOI: 10.1002/anie.202001201 PMID: 32097518 PMC: PMC7318252
pubmed: 32097518
doi: 10.1002/anie.202001201
pmc: PMC7318252
doi:

Substances chimiques

4,4-difluoro-4-bora-3a,4a-diaza-s-indacene 0
Boron Compounds 0
Fluorescent Dyes 0
Intermediate-Conductance Calcium-Activated Potassium Channels 0
KCNN4 protein, human 0
Ligands 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

8277-8284

Informations de copyright

© 2020 The Authors. Published by Wiley-VCH Verlag GmbH & Co. KGaA.

Références

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Auteurs

Kathrin Brömmel (K)

Institute for Pharmaceutical and Medicinal Chemistry, Westphalian Wilhelms-University Münster, Corrensstraße 48, 48149, Münster, Germany.
Cells-in-Motion Interfaculty Center, Westphalian Wilhelms-University Münster, Waldeyerstraße 15, 84149, Münster, Germany.

Sarah Maskri (S)

Institute for Pharmaceutical and Medicinal Chemistry, Westphalian Wilhelms-University Münster, Corrensstraße 48, 48149, Münster, Germany.

Ivan Maisuls (I)

Center for Nanotechnology, Center for Soft Nanoscience, Institute for Inorganic and Analytical Chemistry, Westphalian Wilhelms-University Münster, Heisenbergstraße 11, 48149, Münster, Germany.

Christian Paul Konken (CP)

Department of Nuclear Medicine, University Hospital Münster, Albert-Schweitzer-Campus 1, Building A1, 48149, Münster, Germany.

Marius Rieke (M)

Institute for Physiology II, University Hospital Münster, Robert-Koch-Straße 27b, 48149, Münster, Germany.

Zoltan Pethő (Z)

Institute for Physiology II, University Hospital Münster, Robert-Koch-Straße 27b, 48149, Münster, Germany.

Cristian A Strassert (CA)

Center for Nanotechnology, Center for Soft Nanoscience, Institute for Inorganic and Analytical Chemistry, Westphalian Wilhelms-University Münster, Heisenbergstraße 11, 48149, Münster, Germany.
Cells-in-Motion Interfaculty Center, Westphalian Wilhelms-University Münster, Waldeyerstraße 15, 84149, Münster, Germany.

Oliver Koch (O)

Institute for Pharmaceutical and Medicinal Chemistry, Westphalian Wilhelms-University Münster, Corrensstraße 48, 48149, Münster, Germany.

Albrecht Schwab (A)

Institute for Physiology II, University Hospital Münster, Robert-Koch-Straße 27b, 48149, Münster, Germany.

Bernhard Wünsch (B)

Institute for Pharmaceutical and Medicinal Chemistry, Westphalian Wilhelms-University Münster, Corrensstraße 48, 48149, Münster, Germany.
Cells-in-Motion Interfaculty Center, Westphalian Wilhelms-University Münster, Waldeyerstraße 15, 84149, Münster, Germany.
ORCID: 0000-0002-9030-8417

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Classifications MeSH

questionsmedicales.fr › Cellules › Cellules épithéliales › Cellules A549 › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Phénomènes chimiques › Phénomènes biochimiques › Sites de fixation › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Composés chimiques organiques › Composés du bore › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Technologie, industrie et agriculture › Technologie › Technologie pharmaceutique › Techniques de chimie synthétique › Réaction de cycloaddition › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Actions chimiques et utilisations › Utilisations spécialisées de produits chimiques › Produits chimiques de laboratoire › Indicateurs et réactifs › Luminescents › Colorants fluorescents › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Eucaryotes › Animaux › Chordés › Vertébrés › Mammifères › Eutheria › Primates › Haplorhini › Catarrhini › Hominidae › Humains › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Acides aminés, peptides et protéines › Protéines › Protéines membranaires › Protéines de transport membranaire › Canaux ioniques › Canaux potassiques › Canaux potassiques calcium-dépendants › Canaux potassiques calcium-dépendants de conductance intermédiaire › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Actions chimiques et utilisations › Utilisations spécialisées de produits chimiques › Produits chimiques de laboratoire › Ligands › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Techniques d'investigation › Microscopie de fluorescence › Synthesis of Small-Molecule Fluorescent Probes...
questionsmedicales.fr › Sciences de l'information › Méthodologies informatiques › Simulation numérique › Simulation de dynamique moléculaire › Synthesis of Small-Molecule Fluorescent Probes...