Structure-based discovery of potent and selective melatonin receptor agonists.
GPCR
biased signaling
biochemistry
chemical biology
computational biology
human
melatonin
systems biology
virtual ligand screening
Journal
eLife
ISSN: 2050-084X
Titre abrégé: Elife
Pays: England
ID NLM: 101579614
Informations de publication
Date de publication:
02 03 2020
02 03 2020
Historique:
received:
20
11
2019
accepted:
26
02
2020
pubmed:
3
3
2020
medline:
10
4
2021
entrez:
3
3
2020
Statut:
epublish
Résumé
Melatonin receptors MT
Identifiants
pubmed: 32118583
doi: 10.7554/eLife.53779
pii: 53779
pmc: PMC7080406
doi:
pii:
Substances chimiques
Receptor, Melatonin, MT1
0
Receptor, Melatonin, MT2
0
Receptors, Melatonin
0
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : NIMH NIH HHS
ID : R01 MH112205
Pays : United States
Organisme : NIDDK NIH HHS
ID : U24 DK116195
Pays : United States
Informations de copyright
© 2020, Patel et al.
Déclaration de conflit d'intérêts
NP, XH, JG, LJ, BS, JM, YL, BR, VK No competing interests declared
Références
Chem Biol Drug Des. 2008 Jan;71(1):15-27
pubmed: 18069986
J Med Chem. 2018 Aug 09;61(15):6830-6845
pubmed: 29990431
Neuropharmacology. 2015 Apr;91:142-7
pubmed: 25534555
Curr Med Chem. 2012;19(21):3532-49
pubmed: 22680635
Nature. 2019 May;569(7755):289-292
pubmed: 31019305
J Comput Chem. 2012 Feb 15;33(5):561-72
pubmed: 22170280
Methods Mol Biol. 2012;857:189-205
pubmed: 22323222
Naunyn Schmiedebergs Arch Pharmacol. 2003 Jun;367(6):553-61
pubmed: 12764576
J Med Chem. 2010 Feb 25;53(4):1799-809
pubmed: 20095623
Prog Neurobiol. 2011 Mar;93(3):350-84
pubmed: 21193011
Annu Rev Pharmacol Toxicol. 2016;56:361-83
pubmed: 26514204
Nucleic Acids Res. 2019 Jan 8;47(D1):D1102-D1109
pubmed: 30371825
Behav Brain Res. 2013 Apr 15;243:231-8
pubmed: 23333399
Sci Signal. 2018 Aug 28;11(545):
pubmed: 30154102
J Med Chem. 2010 Apr 8;53(7):2719-40
pubmed: 20131845
Neuron. 1994 Nov;13(5):1177-85
pubmed: 7946354
ACS Chem Neurosci. 2012 Mar 21;3(3):193-203
pubmed: 22860188
Eur J Pharmacol. 2015 Oct 5;764:424-432
pubmed: 26162699
Nucleic Acids Res. 2000 Jan 1;28(1):235-42
pubmed: 10592235
Br J Pharmacol. 2018 Aug;175(16):3263-3280
pubmed: 28707298
Nat Struct Mol Biol. 2019 Jul;26(7):535-544
pubmed: 31270468
Mol Pharmacol. 2013 Dec;84(6):794-807
pubmed: 24021214
Pharmacol Rev. 2019 Apr;71(2):267-315
pubmed: 30914442
Nature. 2019 Feb;566(7743):224-229
pubmed: 30728502
J Med Chem. 2014 Apr 24;57(8):3161-85
pubmed: 24228714
Nature. 2020 Mar;579(7800):609-614
pubmed: 32040955
Cell Tissue Res. 2002 Jul;309(1):127-37
pubmed: 12111543
Nucleic Acids Res. 2017 Jan 4;45(D1):D158-D169
pubmed: 27899622
Nat Rev Endocrinol. 2019 Feb;15(2):105-125
pubmed: 30531911
Nat Struct Mol Biol. 2015 May;22(5):362-9
pubmed: 25895059
N Engl J Med. 1997 Jan 16;336(3):186-95
pubmed: 8988899
J Med Chem. 2017 Apr 13;60(7):3070-3081
pubmed: 28339199
Expert Opin Ther Targets. 2016 Oct;20(10):1209-18
pubmed: 27082492
Endocrine. 2005 Jul;27(2):101-10
pubmed: 16217123
Expert Opin Drug Discov. 2018 Mar;13(3):241-248
pubmed: 29271261
Br J Pharmacol. 2016 Sep;173(18):2702-25
pubmed: 27314810
Science. 2017 Oct 20;358(6361):381-386
pubmed: 29051383
Nat Rev Drug Discov. 2014 Feb;13(2):105-21
pubmed: 24481311
Nature. 2019 May;569(7755):284-288
pubmed: 31019306
Nucleic Acids Res. 2017 Jan 4;45(D1):D945-D954
pubmed: 27899562
Sleep Med. 2006 Jan;7(1):17-24
pubmed: 16309958
J Chem Inf Model. 2012 Jan 23;52(1):1-6
pubmed: 22168315
J Mol Biol. 1994 Jan 21;235(3):983-1002
pubmed: 8289329
Drug Discov Today. 2004 May 15;9(10):430-1
pubmed: 15109945
J Chem Inf Model. 2015 Nov 23;55(11):2324-37
pubmed: 26479676
Neurosci Lett. 2009 Jun 26;457(2):93-6
pubmed: 19429170
Nat Rev Drug Discov. 2010 Aug;9(8):628-42
pubmed: 20577266
Neurol Res. 2017 Jun;39(6):559-565
pubmed: 28460563