Design, Synthesis, Computational, and Preclinical Evaluation of
Animals
Computer Simulation
Glutamic Acid
/ chemistry
Humans
Kallikreins
/ chemistry
Male
Mice
Mice, Inbred BALB C
Neoplasms, Experimental
/ diagnostic imaging
PC-3 Cells
Positron-Emission Tomography
Prostate-Specific Antigen
/ chemistry
Prostatic Neoplasms
/ diagnostic imaging
Pyridones
/ chemistry
Radioactive Tracers
Radiopharmaceuticals
/ chemical synthesis
Titanium
/ chemistry
Urea
/ chemistry
PET
PSMA
titanium-45
Journal
Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009
Informations de publication
Date de publication:
02 Mar 2020
02 Mar 2020
Historique:
received:
31
01
2020
revised:
27
02
2020
accepted:
28
02
2020
entrez:
6
3
2020
pubmed:
7
3
2020
medline:
15
12
2020
Statut:
epublish
Résumé
Despite promising anti-cancer properties in vitro, all titanium-based pharmaceuticals have failed in vivo. Likewise, no target-specific positron emission tomography (PET) tracer based on the radionuclide
Identifiants
pubmed: 32131399
pii: molecules25051104
doi: 10.3390/molecules25051104
pmc: PMC7179113
pii:
doi:
Substances chimiques
Pyridones
0
Radioactive Tracers
0
Radiopharmaceuticals
0
chelidamic acid
138-60-3
Glutamic Acid
3KX376GY7L
Urea
8W8T17847W
Titanium
D1JT611TNE
KLK3 protein, human
EC 3.4.21.-
Kallikreins
EC 3.4.21.-
Prostate-Specific Antigen
EC 3.4.21.77
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Références
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