Alleviating pain with delta opioid receptor agonists: evidence from experimental models.
Delta opioid receptor
G protein-coupled receptors
Pain
Primary afferents
Trafficking
Journal
Journal of neural transmission (Vienna, Austria : 1996)
ISSN: 1435-1463
Titre abrégé: J Neural Transm (Vienna)
Pays: Austria
ID NLM: 9702341
Informations de publication
Date de publication:
04 2020
04 2020
Historique:
received:
19
12
2019
accepted:
06
03
2020
pubmed:
20
3
2020
medline:
16
6
2021
entrez:
20
3
2020
Statut:
ppublish
Résumé
The use of opioids for the relief of pain and headache disorders has been studied for years. Nowadays, particularly because of its ability to produce analgesia in various pain models, delta opioid receptor (DOPr) emerges as a promising target for the development of new pain therapies. Indeed, their potential to avoid the unwanted effects commonly observed with clinically used opioids acting at the mu opioid receptor (MOPr) suggests that DOPr agonists could be a therapeutic option. In this review, we discuss the use of opioids in the management of pain in addition to describing the evidence of the analgesic potency of DOPr agonists in animal models.
Identifiants
pubmed: 32189076
doi: 10.1007/s00702-020-02172-4
pii: 10.1007/s00702-020-02172-4
doi:
Substances chimiques
Analgesics, Opioid
0
Receptors, Opioid, delta
0
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Review
Langues
eng
Sous-ensembles de citation
IM
Pagination
661-672Subventions
Organisme : CIHR
ID : MOP-136871
Pays : Canada
Organisme : CIHR
ID : PJT-162103
Pays : Canada
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