Zerumbone Modulates α
NMDA NR2B
TRPV1
allodynia and hyperalgesia
neuropathic pain
zerumbone
α2A-adrenoceptor
Journal
Frontiers in pharmacology
ISSN: 1663-9812
Titre abrégé: Front Pharmacol
Pays: Switzerland
ID NLM: 101548923
Informations de publication
Date de publication:
2020
2020
Historique:
received:
24
09
2019
accepted:
27
01
2020
entrez:
21
3
2020
pubmed:
21
3
2020
medline:
21
3
2020
Statut:
epublish
Résumé
Zerumbone has shown great potential in various pathophysiological models of diseases, particularly in neuropathic pain conditions. Further understanding the mechanisms of action is important to develop zerumbone as a potential anti-nociceptive agent. Numerous receptors and pathways function to inhibit and modulate transmission of pain signals. Previously, we demonstrated involvement of the serotonergic system in zerumbone's anti-neuropathic effects. The present study was conducted to determine zerumbone's modulatory potential involving noradrenergic, transient receptor potential vanilloid type 1 (TRPV1) and
Identifiants
pubmed: 32194397
doi: 10.3389/fphar.2020.00092
pmc: PMC7064019
doi:
Types de publication
Journal Article
Langues
eng
Pagination
92Informations de copyright
Copyright © 2020 Chia, Izham, Farouk, Sulaiman, Mustafa, Hutchinson and Perimal.
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