The Molecular Control of Calcitonin Receptor Signaling.


Journal

ACS pharmacology & translational science
ISSN: 2575-9108
Titre abrégé: ACS Pharmacol Transl Sci
Pays: United States
ID NLM: 101721411

Informations de publication

Date de publication:
08 Feb 2019
Historique:
received: 14 12 2018
entrez: 29 3 2020
pubmed: 11 1 2019
medline: 11 1 2019
Statut: epublish

Résumé

The calcitonin receptor (CTR) is a class B G protein-coupled receptor (GPCR) that responds to the peptide hormone calcitonin (CT). CTs are clinically approved for the treatment of bone diseases. We previously reported a 4.1 Å structure of the activated CTR bound to salmon CT (sCT) and heterotrimeric Gs protein by cryo-electron microscopy (Liang, Y.-L.,

Identifiants

pubmed: 32219215
doi: 10.1021/acsptsci.8b00056
pmc: PMC7088896
doi:

Types de publication

Journal Article

Langues

eng

Pagination

31-51

Subventions

Organisme : Biotechnology and Biological Sciences Research Council
ID : BB/M006883/1
Pays : United Kingdom

Informations de copyright

Copyright © 2019 American Chemical Society.

Déclaration de conflit d'intérêts

The authors declare no competing financial interest.

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Auteurs

Emma Dal Maso (E)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.

Alisa Glukhova (A)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.

Yue Zhu (Y)

The National Center for Drug Screening and CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.
University of Chinese Academy of Sciences, 19A Yuquan Road, Beijing 100049, China.

Javier Garcia-Nafria (J)

MRC Laboratory of Molecular Biology, Francis Crick Avenue, Cambridge, CB2 0QH, U.K.

Christopher G Tate (CG)

MRC Laboratory of Molecular Biology, Francis Crick Avenue, Cambridge, CB2 0QH, U.K.

Silvia Atanasio (S)

School of Biological Sciences, University of Essex, Wivenhoe Park, Colchester CO4 3SQ, U.K.

Christopher A Reynolds (CA)

School of Biological Sciences, University of Essex, Wivenhoe Park, Colchester CO4 3SQ, U.K.

Erney Ramírez-Aportela (E)

Biocomputing Unit, National Center for Biotechnology (CNB-CSIC), C/Darwin, 3, Campus Universidad Autónoma, 28049 Cantoblanco, Madrid Spain.

Jose-Maria Carazo (JM)

Biocomputing Unit, National Center for Biotechnology (CNB-CSIC), C/Darwin, 3, Campus Universidad Autónoma, 28049 Cantoblanco, Madrid Spain.

Caroline A Hick (CA)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.

Sebastian G B Furness (SGB)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.

Debbie L Hay (DL)

The University of Auckland, School of Biological Sciences, 3 Symonds Street, Auckland 1142, New Zealand.

Yi-Lynn Liang (YL)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.

Laurence J Miller (LJ)

Department of Molecular Pharmacology and Experimental Therapeutics, Mayo Clinic, Scottsdale, Arizona 85259, United States.

Arthur Christopoulos (A)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.

Ming-Wei Wang (MW)

The National Center for Drug Screening and CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.
University of Chinese Academy of Sciences, 19A Yuquan Road, Beijing 100049, China.
School of Pharmacy, Fudan University, Shanghai 201203, China.

Denise Wootten (D)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.
School of Pharmacy, Fudan University, Shanghai 201203, China.

Patrick M Sexton (PM)

Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, Victoria Australia.
School of Pharmacy, Fudan University, Shanghai 201203, China.

Classifications MeSH