Synthesis and Biological Evaluation of Imidazo[2 ,1-

carbonic anhydrase hCA I hCA II hCA IX hCA XII imidazo[2,1-b]thiazole sulfonyl piperazine

Journal

Metabolites
ISSN: 2218-1989
Titre abrégé: Metabolites
Pays: Switzerland
ID NLM: 101578790

Informations de publication

Date de publication:
31 Mar 2020
Historique:
received: 12 03 2020
revised: 27 03 2020
accepted: 28 03 2020
entrez: 5 4 2020
pubmed: 5 4 2020
medline: 5 4 2020
Statut: epublish

Résumé

A novel series of imidazo[2,1-

Identifiants

pubmed: 32244413
pii: metabo10040136
doi: 10.3390/metabo10040136
pmc: PMC7240968
pii:
doi:

Types de publication

Journal Article

Langues

eng

Déclaration de conflit d'intérêts

The authors declare no conflict of interest.

Références

J Enzyme Inhib Med Chem. 2013 Apr;28(2):229-30
pubmed: 23379684
J Med Chem. 2005 Dec 1;48(24):7860-6
pubmed: 16302824
J Enzyme Inhib Med Chem. 2015 Feb;30(1):75-80
pubmed: 24666304
Curr Med Chem Cardiovasc Hematol Agents. 2004 Jan;2(1):49-68
pubmed: 15328829
J Enzyme Inhib Med Chem. 2015;30(4):519-23
pubmed: 25198893
Bioorg Med Chem. 2017 Oct 15;25(20):5726-5732
pubmed: 28887000
Eur J Med Chem. 2017 Jan 27;126:36-51
pubmed: 27744185
J Enzyme Inhib Med Chem. 2016;31(3):345-60
pubmed: 26619898
J Med Chem. 2015 Feb 12;58(3):1494-501
pubmed: 25581127
J Enzyme Inhib Med Chem. 2018 Dec;33(1):303-308
pubmed: 29280407
Biochem J. 2016 Jul 15;473(14):2023-32
pubmed: 27407171
J Med Chem. 2002 Mar 28;45(7):1466-76
pubmed: 11906288
J Med Chem. 2005 Apr 21;48(8):3085-9
pubmed: 15828848
Farmaco. 1993 May;48(5):707-12
pubmed: 8343214
Expert Opin Ther Pat. 2018 Oct;28(10):709-712
pubmed: 30217119
Bioorg Med Chem. 2017 Feb 1;25(3):1286-1293
pubmed: 28065499
Expert Opin Drug Discov. 2019 Nov;14(11):1175-1197
pubmed: 31436118
Eur J Med Chem. 2009 Jul;44(7):2776-81
pubmed: 19203813
Nat Rev Drug Discov. 2008 Feb;7(2):168-81
pubmed: 18167490
Eur J Med Chem. 2011 Jun;46(6):2109-16
pubmed: 21439690
J Enzyme Inhib Med Chem. 2015 Jun;30(3):430-4
pubmed: 25089707
Metabolites. 2018 Mar 21;8(2):
pubmed: 29561812
Expert Opin Drug Discov. 2020 Jun;15(6):671-686
pubmed: 32208982
J Biol Chem. 1971 Apr 25;246(8):2561-73
pubmed: 4994926
ChemMedChem. 2019 Dec 17;14(24):2052-2060
pubmed: 31674147
J Med Chem. 2012 Feb 23;55(4):1721-30
pubmed: 22276570
Expert Opin Drug Discov. 2017 Jan;12(1):61-88
pubmed: 27783541
J Am Chem Soc. 2009 Mar 4;131(8):3057-62
pubmed: 19206230

Auteurs

Kesari Lakshmi Manasa (KL)

Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad-500 037, India.

Sravya Pujitha (S)

Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad-500 037, India.

Aaftaab Sethi (A)

Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad-500 037, India.

Arifuddin Mohammed (A)

Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad-500 037, India.
Department of Chemistry, Anwarul Uloom College, 11-3-918, New Malleypally, Hyderabad-500001, T. S., India (Present Address).

Mallika Alvala (M)

Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad-500 037, India.

Andrea Angeli (A)

Università degli Studi di Firenze, Neurofarba Dept., Sezione di Scienze Farmaceutiche e Nutraceutiche, Via Ugo Schiff 6, 50019 Sesto Fiorentino, Florence, Italy.

Claudiu T Supuran (CT)

Università degli Studi di Firenze, Neurofarba Dept., Sezione di Scienze Farmaceutiche e Nutraceutiche, Via Ugo Schiff 6, 50019 Sesto Fiorentino, Florence, Italy.

Classifications MeSH