A Polyamine-Based Dinitro-Naphthalimide Conjugate as Substrates for Polyamine Transporters Preferentially Accumulates in Cancer Cells and Minimizes Side Effects
cancer
dinitro-naphthalimide conjugate
minimized side-effects
polyamine
polyamine transporter
Journal
Frontiers in chemistry
ISSN: 2296-2646
Titre abrégé: Front Chem
Pays: Switzerland
ID NLM: 101627988
Informations de publication
Date de publication:
2020
2020
Historique:
received:
20
12
2019
accepted:
25
02
2020
entrez:
25
4
2020
pubmed:
25
4
2020
medline:
25
4
2020
Statut:
epublish
Résumé
Naphthalimides, such as amonafide and mitonafide in clinical trials, have been developed as antitumor agents for orthotopic tumor. However, the serious side effects in cancer patients limit their applications. Herein, a new class of polyamine-based naphthalimide conjugates
Identifiants
pubmed: 32328475
doi: 10.3389/fchem.2020.00166
pmc: PMC7160362
doi:
Types de publication
Journal Article
Langues
eng
Pagination
166Informations de copyright
Copyright © 2020 Ma, Li, Li, Yue, Liu, Wang, Xi, Shi, Zhao, Ma, Liu, Guo, Liu, Hou, Wang, Wang, Tian and Xie.
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