TLR7/8 Agonist-Loaded Nanoparticles Augment NK Cell-Mediated Antibody-Based Cancer Immunotherapy.


Journal

Molecular pharmaceutics
ISSN: 1543-8392
Titre abrégé: Mol Pharm
Pays: United States
ID NLM: 101197791

Informations de publication

Date de publication:
01 06 2020
Historique:
pubmed: 10 5 2020
medline: 8 6 2021
entrez: 9 5 2020
Statut: ppublish

Résumé

Activated natural killer (NK) cells can kill malignant tumor cells via granule exocytosis and secretion of IFN-γ, a key regulator of the TH1 response. Thus, mobilization of NK cells can augment cancer immunotherapy, particularly when mediated through antibody-dependent cellular cytotoxicity (ADCC). Stimulation of toll-like receptor (TLR)7/8 activity in dendritic cells promotes pro-inflammatory cytokine secretion and costimulatory molecule upregulation, both of which can potentiate NK cell activation. However, currently available TLR7/8 agonists exhibit unfavorable pharmacokinetics, limiting their

Identifiants

pubmed: 32383885
doi: 10.1021/acs.molpharmaceut.0c00271
doi:

Substances chimiques

Toll-Like Receptor 7 0
Toll-Like Receptor 8 0
Imiquimod P1QW714R7M

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

2109-2124

Auteurs

Hyunjoon Kim (H)

Department of Pharmaceutics, University of Minnesota, Minneapolis, Minnesota 55455, United States.

Vidhi Khanna (V)

Department of Pharmaceutics, University of Minnesota, Minneapolis, Minnesota 55455, United States.

Tamara A Kucaba (TA)

Department of Urology, University of Minnesota, Minneapolis, Minnesota 55455, United States.

Wenqiu Zhang (W)

Department of Pharmaceutics, University of Minnesota, Minneapolis, Minnesota 55455, United States.

Drishti Sehgal (D)

Department of Urology, University of Minnesota, Minneapolis, Minnesota 55455, United States.

David M Ferguson (DM)

Department of Medicinal Chemistry, University of Minnesota, Minneapolis, Minnesota 55455, United States.

Thomas S Griffith (TS)

Department of Urology, University of Minnesota, Minneapolis, Minnesota 55455, United States.
Masonic Cancer Center, University of Minnesota, Minneapolis, Minnesota 55455, United States.
Center for Immunology, University of Minnesota, Minneapolis, Minnesota 55455, United States.
Microbiology, Immunology, and Cancer Biology Graduate Program, University of Minnesota, Minneapolis, Minnesota 55455, United States.

Jayanth Panyam (J)

Department of Pharmaceutics, University of Minnesota, Minneapolis, Minnesota 55455, United States.
Masonic Cancer Center, University of Minnesota, Minneapolis, Minnesota 55455, United States.

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Classifications MeSH