Screening of nanoemulsion components for asenapine maleate using validated RP-HPLC method.


Journal

Annales pharmaceutiques francaises
ISSN: 0003-4509
Titre abrégé: Ann Pharm Fr
Pays: France
ID NLM: 2985176R

Informations de publication

Date de publication:
Sep 2020
Historique:
received: 11 02 2020
revised: 26 04 2020
accepted: 27 04 2020
pubmed: 11 5 2020
medline: 22 6 2021
entrez: 11 5 2020
Statut: ppublish

Résumé

A novel, simple reversed-phase high-performance liquid chromatographic (RP-HPLC) analytical method was developed and validated for the quantitative determination of asenapine from various nanoemulsion components during pre-formulation screening. The developed method was validated according to ICH Q2 (R1) guidelines. The developed and validated method was precisely and accurately quantified asenapine in various oils, surfactants and co-surfactants. The separation of asenapine was carried out on Hypersil BDS C18, 250×4.6mm, 5μm particle size column using methanol: acetonitrile (90:10) as mobile phase with a flow rate of 1mL.min

Identifiants

pubmed: 32387177
pii: S0003-4509(20)30053-5
doi: 10.1016/j.pharma.2020.04.005
pii:
doi:

Substances chimiques

Dibenzocycloheptenes 0
Emulsions 0
Indicators and Reagents 0
Oils 0
Surface-Active Agents 0
asenapine JKZ19V908O

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

379-387

Informations de copyright

Copyright © 2020 Académie Nationale de Pharmacie. Published by Elsevier Masson SAS. All rights reserved.

Auteurs

S A Kumbhar (SA)

School of Pharmaceutical Sciences, Jaipur National University, 302017 Jaipur, Rajasthan, India; Department of Pharmaceutics, STES's Sinhgad Institute of Pharmacy (Affiliated to Savitribai Phule Pune University), India.

C R Kokare (CR)

Department of Pharmaceutics, STES's Sinhgad Institute of Pharmacy (Affiliated to Savitribai Phule Pune University), India.

B Shrivastava (B)

School of Pharmaceutical Sciences, Jaipur National University, 302017 Jaipur, Rajasthan, India. Electronic address: director_pharmacy@jnujaipur.ac.in.

B Gorain (B)

School of Pharmacy, Faculty of Health and Medical Sciences, Taylor's University, 47500 Subang Jaya, Selangor, Malaysia. Electronic address: bapi.gorain@taylors.edu.my.

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