Pharmacologic TWIK-Related Acid-Sensitive K+ Channel (TASK-1) Potassium Channel Inhibitor A293 Facilitates Acute Cardioversion of Paroxysmal Atrial Fibrillation in a Porcine Large Animal Model.
Animals
Anti-Arrhythmia Agents
/ pharmacology
Atrial Fibrillation
/ diagnosis
Disease Models, Animal
Electrocardiography
Electrophysiologic Techniques, Cardiac
Female
Heart Rate
/ drug effects
Humans
Male
Membrane Potentials
/ drug effects
Molecular Docking Simulation
Myocytes, Cardiac
/ drug effects
Nerve Tissue Proteins
/ antagonists & inhibitors
Potassium Channel Blockers
/ pharmacology
Potassium Channels, Tandem Pore Domain
/ antagonists & inhibitors
Proof of Concept Study
Refractory Period, Electrophysiological
/ drug effects
Sulfonamides
/ pharmacology
Sus scrofa
Time Factors
Xenopus laevis
ortho-Aminobenzoates
/ pharmacology
A293
K2P3.1
TASK‐1
antiarrhythmic pharmacotherapy
atrial fibrillation
cardioversion
Journal
Journal of the American Heart Association
ISSN: 2047-9980
Titre abrégé: J Am Heart Assoc
Pays: England
ID NLM: 101580524
Informations de publication
Date de publication:
18 05 2020
18 05 2020
Historique:
pubmed:
12
5
2020
medline:
10
3
2021
entrez:
12
5
2020
Statut:
ppublish
Résumé
Background The tandem of P domains in a weak inward rectifying K+ channel (TWIK)-related acid-sensitive K
Identifiants
pubmed: 32390491
doi: 10.1161/JAHA.119.015751
pmc: PMC7660874
doi:
Substances chimiques
2-(butane-1-sulfonylamino)-N-(1-(6-methoxypyridin-3-yl)propyl)benzamide
0
Anti-Arrhythmia Agents
0
Nerve Tissue Proteins
0
Potassium Channel Blockers
0
Potassium Channels, Tandem Pore Domain
0
Sulfonamides
0
ortho-Aminobenzoates
0
potassium channel subfamily K member 3
1HQ3YCN4GS
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Video-Audio Media
Langues
eng
Sous-ensembles de citation
IM
Pagination
e015751Références
Cell Physiol Biochem. 2011;28(4):613-24
pubmed: 22178873
J Comput Chem. 2009 Dec;30(16):2785-91
pubmed: 19399780
Circ Res. 2006 Apr 28;98(8):1072-80
pubmed: 16574908
Electrophoresis. 2009 Jun;30 Suppl 1:S162-73
pubmed: 19517507
Am J Physiol. 1998 Jul;275(1):H301-21
pubmed: 9688927
Europace. 2016 Nov;18(11):1609-1678
pubmed: 27567465
J Comput Chem. 2010 Jan 30;31(2):455-61
pubmed: 19499576
Nucleic Acids Res. 2014 Jul;42(Web Server issue):W252-8
pubmed: 24782522
Front Med (Lausanne). 2017 Oct 23;4:177
pubmed: 29109948
Circulation. 2016 Apr 5;133(14):1371-85
pubmed: 26912814
Pflugers Arch. 2015 May;467(5):1081-90
pubmed: 25511502
Eur Respir J. 2001 Jul;18(1):221-7
pubmed: 11510795
N Engl J Med. 2013 Jul 25;369(4):351-361
pubmed: 23883380
Pflugers Arch. 2015 May;467(5):1001-11
pubmed: 25476848
Front Physiol. 2013 Jan 04;3:487
pubmed: 23316167
PLoS One. 2017 Mar 16;12(3):e0174071
pubmed: 28301582
Clin Sci (Lond). 2016 May;130(9):643-50
pubmed: 26993052
Heart Rhythm. 2014 Oct;11(10):1798-805
pubmed: 24952150
Circulation. 2015 Jul 14;132(2):82-92
pubmed: 25951834
Cell Physiol Biochem. 2019;52(5):1223-1235
pubmed: 31001961
Mol Biol Cell. 2019 Jun 1;30(12):1425-1436
pubmed: 30969900
J Am Coll Cardiol. 2019 Jul 9;74(1):104-132
pubmed: 30703431
Cardiovasc Res. 2007 Jul 1;75(1):59-68
pubmed: 17389142
Circulation. 2016 Mar 15;133(11):e439
pubmed: 26976922
J Mol Cell Cardiol. 2015 Apr;81:71-80
pubmed: 25655935
Basic Res Cardiol. 2018 Jun 7;113(4):27
pubmed: 29881975
Hypertension. 2011 Oct;58(4):672-8
pubmed: 21876070
Nat Rev Cardiol. 2016 Apr;13(4):230-7
pubmed: 26701216
Europace. 2012 Nov;14 Suppl 5:v17-v24
pubmed: 23104910
Nucleic Acids Res. 2009 Jan;37(Database issue):D387-92
pubmed: 18931379
J Cardiovasc Pharmacol. 2007 Apr;49(4):197-206
pubmed: 17438404
Nat Rev Neurosci. 2001 Mar;2(3):175-84
pubmed: 11256078
Bioinformatics. 2006 Jan 15;22(2):195-201
pubmed: 16301204
Eur Heart J. 2017 Jun 7;38(22):1764-1774
pubmed: 28057773
Trends Pharmacol Sci. 2008 Nov;29(11):566-75
pubmed: 18823665
Am J Physiol Cell Physiol. 2007 Oct;293(4):C1319-26
pubmed: 17699638
Naunyn Schmiedebergs Arch Pharmacol. 2010 Mar;381(3):187-93
pubmed: 20082192
Circ Arrhythm Electrophysiol. 2019 Sep;12(9):e007465
pubmed: 31514528
J Am Heart Assoc. 2020 May 18;9(10):e015751
pubmed: 32390491
Nature. 2017 Jul 20;547(7663):364-368
pubmed: 28693035
Prog Biophys Mol Biol. 2008 Jan-Apr;96(1-3):3-18
pubmed: 17900668
Eur J Pharmacol. 2013 Dec 5;721(1-3):237-48
pubmed: 24070813