Hydroxychloroquine in Coronavirus Disease 2019 Patients: What Still Needs to Be Known About the Kinetics.

COVID-19 dosage regimens drug monitoring hydroxychloroquine population pharmacokinetic modeling

Journal

Clinical infectious diseases : an official publication of the Infectious Diseases Society of America
ISSN: 1537-6591
Titre abrégé: Clin Infect Dis
Pays: United States
ID NLM: 9203213

Informations de publication

Date de publication:
31 12 2020
Historique:
received: 10 04 2020
accepted: 07 05 2020
pubmed: 12 5 2020
medline: 7 1 2021
entrez: 12 5 2020
Statut: ppublish

Résumé

Different dosage regimens of hydroxychloroquine are used to manage coronavirus disease 2019 (COVID-19) patients, without information on the pharmacokinetics in this population. Blood samples (n = 101) were collected from 57 COVID-19 patients for 7 days, and concentrations were compared with simulated kinetic profiles. Hydroxychloroquine exposure is low and cannot be predicted by other populations.

Identifiants

pubmed: 32392332
pii: 5835847
doi: 10.1093/cid/ciaa558
pmc: PMC7239205
doi:

Substances chimiques

Antiviral Agents 0
Hydroxychloroquine 4QWG6N8QKH

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

2962-2964

Informations de copyright

© The Author(s) 2020. Published by Oxford University Press for the Infectious Diseases Society of America. All rights reserved. For permissions, e-mail: journals.permissions@oup.com.

Auteurs

Guillaume Martin-Blondel (G)

Service des Maladies Infectieuses et Tropicales, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Stéphanie Ruiz (S)

Service de Réanimation - Rangueil, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Marlène Murris (M)

Service de Pneumologie - CRCM, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Stanilas Faguer (S)

Pôle de Néphrologie et Transplantation d'Organes, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Véronigue Duhalde (V)

Pôle Pharmacie, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Frédéric Eyvrard (F)

Pôle Pharmacie, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Jacques Izopet (J)

Laboratoire de Virologie, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Jean-Michel Mansuy (JM)

Laboratoire de Virologie, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Yves Rolland (Y)

Pôle de Gériatrie, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Karen Delavigne (K)

Service d'Hématologie, IUCT-Oncopole, Toulouse, France.

Rosine Guimbaud (R)

Pôle des Maladies de l'Appareil Digestif, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Grégory Pugnet (G)

Service de Médecine Interne, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Jean-Marie Conil (JM)

Service de Réanimation - Rangueil, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Bernard Georges (B)

Service de Réanimation - Rangueil, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Pierre Delobel (P)

Service des Maladies Infectieuses et Tropicales, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Vincent Minville (V)

Service de Réanimation - Rangueil, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Stein Silva Sifontes (S)

Service de Réanimation - Purpan, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

Didier Concordet (D)

UMR INTHERES, INRA-ENVT, Toulouse, France.

Peggy Gandia (P)

UMR INTHERES, INRA-ENVT, Toulouse, France.
Laboratoire de Pharmacocinétique et Toxicologie, Centre Hospitalo-Universitaire de Toulouse, Toulouse, France.

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Classifications MeSH