Prioritization of Anti-SARS-Cov-2 Drug Repurposing Opportunities Based on Plasma and Target Site Concentrations Derived from their Established Human Pharmacokinetics.


Journal

Clinical pharmacology and therapeutics
ISSN: 1532-6535
Titre abrégé: Clin Pharmacol Ther
Pays: United States
ID NLM: 0372741

Informations de publication

Date de publication:
10 2020
Historique:
received: 24 04 2020
accepted: 18 05 2020
pubmed: 22 5 2020
medline: 30 9 2020
entrez: 22 5 2020
Statut: ppublish

Résumé

There is a rapidly expanding literature on the in vitro antiviral activity of drugs that may be repurposed for therapy or chemoprophylaxis against severe acute respiratory syndrome-coronavirus 2 (SARS-CoV-2). However, this has not been accompanied by a comprehensive evaluation of the target plasma and lung concentrations of these drugs following approved dosing in humans. Accordingly, concentration 90% (EC

Identifiants

pubmed: 32438446
doi: 10.1002/cpt.1909
pmc: PMC7280633
doi:

Substances chimiques

Antiviral Agents 0

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't Review

Langues

eng

Sous-ensembles de citation

IM

Pagination

775-790

Subventions

Organisme : Medical Research Council
ID : MC_PC_17167
Pays : United Kingdom
Organisme : NIAID NIH HHS
ID : R24 AI118397
Pays : United States
Organisme : NIAID NIH HHS
ID : R01 AI134091
Pays : United States

Commentaires et corrections

Type : ErratumIn

Informations de copyright

© 2020 The Authors. Clinical Pharmacology & Therapeutics published by Wiley Periodicals LLC on behalf of American Society for Clinical Pharmacology and Therapeutics.

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Auteurs

Usman Arshad (U)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Henry Pertinez (H)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Helen Box (H)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Lee Tatham (L)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Rajith K R Rajoli (RKR)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Paul Curley (P)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Megan Neary (M)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Joanne Sharp (J)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Neill J Liptrott (NJ)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Anthony Valentijn (A)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Christopher David (C)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Steve P Rannard (SP)

Department of Chemistry, University of Liverpool, Liverpool, UK.

Paul M O'Neill (PM)

Department of Chemistry, University of Liverpool, Liverpool, UK.

Ghaith Aljayyoussi (G)

Department of Tropical Disease Biology, Liverpool School of Tropical Medicine, Centre for Drugs and Diagnostics, Liverpool, UK.

Shaun H Pennington (SH)

Department of Tropical Disease Biology, Liverpool School of Tropical Medicine, Centre for Drugs and Diagnostics, Liverpool, UK.

Stephen A Ward (SA)

Department of Tropical Disease Biology, Liverpool School of Tropical Medicine, Centre for Drugs and Diagnostics, Liverpool, UK.

Andrew Hill (A)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

David J Back (DJ)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Saye H Khoo (SH)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

Patrick G Bray (PG)

Pat Bray Electrical, Wigan, UK.

Giancarlo A Biagini (GA)

Department of Tropical Disease Biology, Liverpool School of Tropical Medicine, Centre for Drugs and Diagnostics, Liverpool, UK.

Andrew Owen (A)

Department of Molecular and Clinical Pharmacology, Materials Innovation Factory, University of Liverpool, Liverpool, UK.

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