The Relationship Between Dipeptidyl Peptidase-4 Inhibitor Usage and Asymptomatic Amylase Lipase Increment in Type 2 Diabetes Mellitus Patients.

Oral antidiabetics amylase dipeptidyl peptidase-4 inhibitors lipase

Journal

Turkish journal of pharmaceutical sciences
ISSN: 2148-6247
Titre abrégé: Turk J Pharm Sci
Pays: Turkey
ID NLM: 101717890

Informations de publication

Date de publication:
Feb 2020
Historique:
received: 21 08 2018
accepted: 25 10 2018
entrez: 27 5 2020
pubmed: 27 5 2020
medline: 27 5 2020
Statut: ppublish

Résumé

In different studies, it has been shown that the use of dipeptidyl peptidase-4 (DPP-4) inhibitors (DPP-4 inh) does not increase the risk of pancreatitis or pancreatic cancer. Although the number of studies involving clinical pancreatitis clinics is sufficient, the number of studies involving clinical non-pancreatitis hyperamylasemia is rare. The aim of the study was to investigate the relationship between DPP-4 inh usage and amylase and lipase increment without clinical pancreatitis symptoms. Eighty-seven patients who met the inclusion criteria were enrolled. The patients were divided into 3 groups according to their use of saxagliptin, sitagliptin, or vildagliptin. All patients included in the study were receiving metformin at a dose of 2 g/day. Fasting blood glucose, postprandial blood glucose, HbA1C, serum creatinine, ALT, amylase, and lipase results were recorded at the beginning of treatment and at the end of 3 months. There was an increase in all groups in terms of amylase and lipase values but there was no significant difference between the groups in terms of increase (p>0.05) There was no statistically significant increase in the saxagliptin and vildagliptin groups (p>0.05) when the baseline and 3-month values of lipase and amylase increase were examined. However, there was a statistically significant increase in amylase and lipase in the sitagliptin group (p<0.05). The use of DPP-4 inh can increase amylase and lipase levels without clinical findings of acute pancreatitis in the patient. DPP-4 inh should be used with caution in patients at risk for pancreatitis and pancreatic cancer. Patients using DPP-4 inh, especially sitagliptin, should be evaluated carefully for pancreatitis risk factors.

Identifiants

pubmed: 32454763
doi: 10.4274/tjps.galenos.2018.83788
pii: 20273
pmc: PMC7227863
doi:

Types de publication

Journal Article

Langues

eng

Pagination

68-73

Informations de copyright

©Copyright 2020 Turk J Pharm Sci, Published by Galenos Publishing House.

Déclaration de conflit d'intérêts

Conflicts of interest: No conflict of interest was declared by the authors.

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Auteurs

Zeynel Abidin Sayiner (ZA)

Gaziantep University, School of Medicine, Department of Endocrinology and Metabolism, Gaziantep, Turkey.

Gamze Inan Demiroğlu (G)

Gaziantep University, School of Medicine, Department of Internal Medicine, Gaziantep, Turkey.

Ersin Akarsu (E)

Gaziantep University, School of Medicine, Department of Endocrinology and Metabolism, Gaziantep, Turkey.

Mustafa Araz (M)

Gaziantep University, School of Medicine, Department of Endocrinology and Metabolism, Gaziantep, Turkey.

Classifications MeSH