Parabens inhibit hNa

Anticonvulsant drugs Benzylparaben Benzylparaben (CID:7180) Butylparaben (CID:7184) Ethylparaben (CID:8434) Methylparaben (CID:7456) Propylparaben Propylparaben (CID:7175) hNa(V) 1.2 sodium channels

Journal

Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie
ISSN: 1950-6007
Titre abrégé: Biomed Pharmacother
Pays: France
ID NLM: 8213295

Informations de publication

Date de publication:
Aug 2020
Historique:
received: 05 02 2020
revised: 27 04 2020
accepted: 10 05 2020
pubmed: 2 6 2020
medline: 27 2 2021
entrez: 2 6 2020
Statut: ppublish

Résumé

Propylparaben, a commonly used antimicrobial preservative, has been reported as an anticonvulsant agent targeting neuronal Na

Identifiants

pubmed: 32480218
pii: S0753-3322(20)30442-X
doi: 10.1016/j.biopha.2020.110250
pii:
doi:

Substances chimiques

NAV1.2 Voltage-Gated Sodium Channel 0
Parabens 0
SCN2A protein, human 0
Voltage-Gated Sodium Channel Blockers 0
butylparaben 3QPI1U3FV8
benzylparaben 8Y41DYV4VG
propylparaben Z8IX2SC1OH

Types de publication

Comparative Study Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

110250

Informations de copyright

Copyright © 2020. Published by Elsevier Masson SAS.

Déclaration de conflit d'intérêts

Declaration of Competing Interest The authors declare no conflicts of interest.

Auteurs

Andrea Enrique (A)

Instituto de Estudios Inmunológicos y Fisiopatológicos (IIFP), UNLP, CONICET, asociado CIC PBA, Facultad de Ciencias Exactas, La Plata, Argentina. Electronic address: andreaenrique@biol.unlp.edu.ar.

Pedro Martín (P)

Instituto de Estudios Inmunológicos y Fisiopatológicos (IIFP), UNLP, CONICET, asociado CIC PBA, Facultad de Ciencias Exactas, La Plata, Argentina. Electronic address: pedromartin@biol.unlp.edu.ar.

María Laura Sbaraglini (ML)

Laboratorio de Investigación y Desarrollo de Bioactivos (LIDeB), Departamento de Ciencias Biológicas, Facultad de Ciencias Exactas, Universidad Nacional de La Plata, La Plata, Argentina. Electronic address: mariasbara@gmail.com.

Alan Talevi (A)

Laboratorio de Investigación y Desarrollo de Bioactivos (LIDeB), Departamento de Ciencias Biológicas, Facultad de Ciencias Exactas, Universidad Nacional de La Plata, La Plata, Argentina. Electronic address: atalevi@biol.unlp.edu.ar.

Verónica Milesi (V)

Instituto de Estudios Inmunológicos y Fisiopatológicos (IIFP), UNLP, CONICET, asociado CIC PBA, Facultad de Ciencias Exactas, La Plata, Argentina. Electronic address: veronica@biol.unlp.edu.ar.

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Classifications MeSH