Silencing of spontaneous activity at α4β1/3δ GABA
Journal
British journal of pharmacology
ISSN: 1476-5381
Titre abrégé: Br J Pharmacol
Pays: England
ID NLM: 7502536
Informations de publication
Date de publication:
09 2020
09 2020
Historique:
received:
27
05
2019
revised:
10
05
2020
accepted:
14
05
2020
pubmed:
3
6
2020
medline:
22
6
2021
entrez:
3
6
2020
Statut:
ppublish
Résumé
The δ-subunit-containing GABA Whole-cell electrophysiological recordings of adult male rat and mouse hippocampal DGGCs were used to characterize known agonists and antagonists at δ-subunit-containing GABA Recordings at either 24°C or 34°C, including the PKC autoinhibitory peptide (19-36) intracellularly, removed spontaneous gating by GABA Kinase activity infers spontaneous gating in α
Sections du résumé
BACKGROUND AND PURPOSE
The δ-subunit-containing GABA
EXPERIMENTAL APPROACH
Whole-cell electrophysiological recordings of adult male rat and mouse hippocampal DGGCs were used to characterize known agonists and antagonists at δ-subunit-containing GABA
KEY RESULTS
Recordings at either 24°C or 34°C, including the PKC autoinhibitory peptide (19-36) intracellularly, removed spontaneous gating by GABA
CONCLUSION AND IMPLICATIONS
Kinase activity infers spontaneous gating in α
Identifiants
pubmed: 32484592
doi: 10.1111/bph.15146
pmc: PMC7429488
doi:
Substances chimiques
Ligands
0
Receptors, GABA-A
0
gamma-Aminobutyric Acid
56-12-2
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
3975-3990Subventions
Organisme : Lundbeck Foundation
ID : R133-A12270
Organisme : Lundbeck Foundation
ID : R192-2015-666
Organisme : Lundbeck Foundation
ID : R230-2016-2562
Informations de copyright
© 2020 The British Pharmacological Society.
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