Discovery of Dihydropyrrolo[1,2-


Journal

Journal of medicinal chemistry
ISSN: 1520-4804
Titre abrégé: J Med Chem
Pays: United States
ID NLM: 9716531

Informations de publication

Date de publication:
23 07 2020
Historique:
pubmed: 17 6 2020
medline: 15 12 2020
entrez: 16 6 2020
Statut: ppublish

Résumé

The

Identifiants

pubmed: 32538088
doi: 10.1021/acs.jmedchem.9b01733
pmc: PMC7961853
mid: NIHMS1678890
doi:

Substances chimiques

Isoquinolines 0
NR2C NMDA receptor 0
NR2D NMDA receptor 0
Pyrazines 0
Pyrroles 0
Receptors, N-Methyl-D-Aspartate 0

Types de publication

Journal Article Research Support, N.I.H., Extramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

7569-7600

Subventions

Organisme : NINDS NIH HHS
ID : R01 NS065371
Pays : United States
Organisme : NINDS NIH HHS
ID : R35 NS111619
Pays : United States

Références

Nature. 1984 Feb 2-8;307(5950):462-5
pubmed: 6320006
Trends Neurosci. 2008 May;31(5):234-42
pubmed: 18395805
Nature. 1993 Jan 7;361(6407):31-9
pubmed: 8421494
Ann N Y Acad Sci. 2003 Nov;1003:318-27
pubmed: 14684455
Nature. 1984 May 17-23;309(5965):261-3
pubmed: 6325946
Nature. 2012 Apr 29;486(7402):256-60
pubmed: 22699619
Neuron. 2016 Mar 2;89(5):983-99
pubmed: 26875626
J Physiol. 2005 Mar 1;563(Pt 2):345-58
pubmed: 15649985
Neurotherapeutics. 2009 Oct;6(4):693-702
pubmed: 19789073
J Comp Neurol. 1994 Sep 1;347(1):150-60
pubmed: 7798379
Nat Rev Neurosci. 2013 Jun;14(6):383-400
pubmed: 23686171
N Engl J Med. 2003 Apr 3;348(14):1333-41
pubmed: 12672860
J Neurosci. 2013 Oct 30;33(44):17290-300
pubmed: 24174662
Nat Commun. 2010 Oct 05;1:90
pubmed: 20981015
J Neurosci. 2008 Apr 2;28(14):3623-30
pubmed: 18385321
PLoS One. 2009 Oct 19;4(10):e7486
pubmed: 19838302
Psychiatr Genet. 2005 Sep;15(3):215-21
pubmed: 16094258
J Med Chem. 2018 Aug 9;61(15):6401-6420
pubmed: 29589935
Neuropsychopharmacology. 2014 Feb;39(3):625-37
pubmed: 24008353
Eur Arch Psychiatry Clin Neurosci. 2010 Mar;260(2):101-11
pubmed: 19856012
J Med Chem. 2016 Mar 24;59(6):2760-79
pubmed: 26919761
ACS Med Chem Lett. 2016 Oct 31;8(1):84-89
pubmed: 28105280
Neuropsychopharmacology. 2012 Jan;37(1):4-15
pubmed: 21956446
J Physiol. 2008 Jan 1;586(1):227-45
pubmed: 17962328
J Neurophysiol. 1998 Feb;79(2):555-66
pubmed: 9463421
J Physiol. 2020 Feb;598(4):633-650
pubmed: 31876958
Nat Neurosci. 2012 Jan 15;15(3):406-13, S1-2
pubmed: 22246434
Neuropharmacology. 2001 Mar;40(4):491-500
pubmed: 11249958
Mol Pharmacol. 2016 Dec;90(6):689-702
pubmed: 27625038
J Neurosci. 1998 Dec 1;18(23):9727-32
pubmed: 9822733
J Physiol. 2012 Aug 15;590(16):3857-75
pubmed: 22641781
Nature. 2012 Jun 13;486(7402):261-5
pubmed: 22699620
Brain. 2012 May;135(Pt 5):1606-21
pubmed: 22544902
CNS Neurosci Ther. 2018 Feb;24(2):144-153
pubmed: 29230960
J Physiol. 1998 Jul 1;510 ( Pt 1):1-18
pubmed: 9625862
Nat Neurosci. 2003 Feb;6(2):144-52
pubmed: 12524545
Pharmacol Rev. 2010 Sep;62(3):405-96
pubmed: 20716669
J Physiol. 2008 Sep 15;586(18):4425-39
pubmed: 18635641
Neuron. 1994 Mar;12(3):529-40
pubmed: 7512349
NeuroRx. 2004 Jan;1(1):101-10
pubmed: 15717010
J Pharmacol Exp Ther. 2016 Mar;356(3):702-11
pubmed: 26675679
J Physiol. 2007 May 15;581(Pt 1):107-28
pubmed: 17303642
Sci Rep. 2019 May 20;9(1):7572
pubmed: 31110197
ACS Med Chem Lett. 2013 Mar 12;4(4):419-22
pubmed: 24900687
J Neurosci. 2016 Nov 2;36(44):11151-11157
pubmed: 27807157
J Med Chem. 2014 Mar 27;57(6):2334-56
pubmed: 24512267
Biol Psychiatry. 2010 Jan 15;67(2):139-45
pubmed: 19897179
Schizophr Bull. 2012 Sep;38(5):920-6
pubmed: 22987850
Ann Neurol. 1988 Oct;24(4):543-51
pubmed: 2853604
Neuropharmacology. 2017 Jul 15;121:204-218
pubmed: 28457974
Front Cell Neurosci. 2015 Mar 25;9:95
pubmed: 25859181
J Med Chem. 2000 Jun 29;43(13):2575-85
pubmed: 10891117
J Psychiatr Res. 1999 Nov-Dec;33(6):523-33
pubmed: 10628529
Brain Res Bull. 2001 Jul 15;55(5):631-40
pubmed: 11576760
J Neurosci. 2010 Apr 28;30(17):5866-75
pubmed: 20427647
Pharmacol Ther. 2004 May;102(2):155-74
pubmed: 15163596
Bioorg Med Chem Lett. 2009 Oct 1;19(19):5560-4
pubmed: 19720530
Nature. 1986 May 29-Jun 4;321(6069):519-22
pubmed: 3012362
J Med Chem. 2013 Jul 11;56(13):5351-81
pubmed: 23627311
J Neurosci. 1998 Jun 1;18(11):4177-88
pubmed: 9592097
Mol Pharmacol. 2014 Nov;86(5):548-60
pubmed: 25205677
Biol Psychiatry. 2000 Feb 15;47(4):351-4
pubmed: 10686270
Mol Pharmacol. 2007 Oct;72(4):907-20
pubmed: 17622578
Behav Pharmacol. 2020 Sep;31(6):524-534
pubmed: 31860561
Science. 1984 Nov 16;226(4676):850-2
pubmed: 6093256
J Med Chem. 2017 Jul 13;60(13):5556-5585
pubmed: 28586221
Expert Opin Ther Pat. 2012 Nov;22(11):1337-52
pubmed: 23009122
Neuroreport. 1992 Dec;3(12):1138-40
pubmed: 1493227
J Physiol. 2005 Nov 15;569(Pt 1):209-21
pubmed: 16141268
Nature. 1999 Sep 2;401(6748):63-9
pubmed: 10485705
Curr Opin Physiol. 2018 Apr;2:27-35
pubmed: 29756080
Neuropharmacology. 2013 Jan;64:13-26
pubmed: 22796429
Expert Opin Ther Pat. 2014 Dec;24(12):1349-66
pubmed: 25351527
Schizophr Bull. 2012 Sep;38(5):950-7
pubmed: 22355184
Expert Opin Drug Discov. 2010 Mar;5(3):235-48
pubmed: 22823020
Lancet Neurol. 2008 Dec;7(12):1091-8
pubmed: 18851928
Pharm Res. 2011 May;28(5):962-77
pubmed: 21052797
Trends Neurosci. 2010 Nov;33(11):513-23
pubmed: 20850189

Auteurs

Matthew P Epplin (MP)

Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.

Ayush Mohan (A)

Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.

Lynnea D Harris (LD)

Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.

Zongjian Zhu (Z)

Department of Pharmacology and Chemical Biology, Emory University, 1510 Clifton Road, Atlanta, Georgia 30322, United States.

Katie L Strong (KL)

Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.

John Bacsa (J)

Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.

Phuong Le (P)

Department of Pharmacology and Chemical Biology, Emory University, 1510 Clifton Road, Atlanta, Georgia 30322, United States.

David S Menaldino (DS)

Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.

Stephen F Traynelis (SF)

Department of Pharmacology and Chemical Biology, Emory University, 1510 Clifton Road, Atlanta, Georgia 30322, United States.

Dennis C Liotta (DC)

Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.

Articles similaires

Smoking Cessation and Incident Cardiovascular Disease.

Jun Hwan Cho, Seung Yong Shin, Hoseob Kim et al.
1.00
Humans Male Smoking Cessation Cardiovascular Diseases Female
Humans United States Aged Cross-Sectional Studies Medicare Part C
1.00
Humans Yoga Low Back Pain Female Male
Humans Meals Time Factors Female Adult

Classifications MeSH