Pharmacokinetic-Pharmacodynamic Target Attainment Analyses To Support Dose Selection for ME1100, an Arbekacin Inhalation Solution.


Journal

Antimicrobial agents and chemotherapy
ISSN: 1098-6596
Titre abrégé: Antimicrob Agents Chemother
Pays: United States
ID NLM: 0315061

Informations de publication

Date de publication:
21 09 2020
Historique:
received: 19 12 2019
accepted: 03 07 2020
pubmed: 15 7 2020
medline: 22 6 2021
entrez: 15 7 2020
Statut: epublish

Résumé

ME1100 (arbekacin inhalation solution) is an inhaled aminoglycoside that is being developed to treat patients with hospital-acquired and ventilator-associated bacterial pneumonia (HABP and VABP, respectively). Pharmacokinetic-pharmacodynamic (PK-PD) target attainment analyses were undertaken to evaluate ME1100 regimens for the treatment of patients with HABP/VABP. The data used included a population pharmacokinetic (PPK) 4-compartment model with 1st-order elimination, nonclinical PK-PD targets from one-compartment

Identifiants

pubmed: 32661000
pii: AAC.02367-19
doi: 10.1128/AAC.02367-19
pmc: PMC7508573
pii:
doi:

Substances chimiques

Anti-Bacterial Agents 0
Dibekacin 45ZFO9E525
arbekacin G7V6SLI20L

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Informations de copyright

Copyright © 2020 American Society for Microbiology.

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Auteurs

Sujata M Bhavnani (SM)

Institute for Clinical Pharmacodynamics, Inc., Schenectady, New York, USA sbhavnani@icpd.com.

Jeffrey P Hammel (JP)

Institute for Clinical Pharmacodynamics, Inc., Schenectady, New York, USA.

Elizabeth A Lakota (EA)

Institute for Clinical Pharmacodynamics, Inc., Schenectady, New York, USA.

M Courtney Safir (MC)

Institute for Clinical Pharmacodynamics, Inc., Schenectady, New York, USA.

Brian D VanScoy (BD)

Institute for Clinical Pharmacodynamics, Inc., Schenectady, New York, USA.

Yu Nagira (Y)

Meiji Seika Pharma Co., Ltd., Tokyo, Japan.

Christopher M Rubino (CM)

Institute for Clinical Pharmacodynamics, Inc., Schenectady, New York, USA.

Nobuo Sato (N)

Meiji Seika Pharma Co., Ltd., Tokyo, Japan.

Tomokazu Koresawa (T)

Meiji Seika Pharma Co., Ltd., Tokyo, Japan.

Kenichiro Kondo (K)

Meiji Seika Pharma Co., Ltd., Tokyo, Japan.

Paul G Ambrose (PG)

Institute for Clinical Pharmacodynamics, Inc., Schenectady, New York, USA.

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Classifications MeSH