Targeting Discoidin Domain Receptor 1 (DDR1) Signaling and Its Crosstalk with β
ATP Binding Cassette Transporter, Subfamily G, Member 2
/ antagonists & inhibitors
Adenocarcinoma
/ drug therapy
Biological Transport
/ drug effects
Breast Neoplasms
/ drug therapy
Cell Adhesion
/ drug effects
Cell Line, Tumor
Collagen Type I
/ metabolism
Discoidin Domain Receptor 1
/ antagonists & inhibitors
Doxorubicin
/ metabolism
Drug Resistance, Neoplasm
/ physiology
ErbB Receptors
/ biosynthesis
Focal Adhesion Kinase 1
/ metabolism
Gefitinib
/ pharmacology
Gene Expression Regulation, Neoplastic
/ drug effects
Gene Knockdown Techniques
Humans
Indazoles
/ pharmacology
Integrin beta1
/ genetics
Integrin beta4
/ biosynthesis
MAP Kinase Signaling System
/ drug effects
MCF-7 Cells
Mitogen-Activated Protein Kinase 1
/ antagonists & inhibitors
Mitogen-Activated Protein Kinase 3
/ antagonists & inhibitors
Mitoxantrone
/ metabolism
Neoplasm Proteins
/ antagonists & inhibitors
Piperazines
/ pharmacology
Tumor Microenvironment
/ drug effects
ABC transporter
DDR1
EGFR
MAPK
breast cancer
chemoresistance
collagen
integrin
Journal
International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791
Informations de publication
Date de publication:
13 Jul 2020
13 Jul 2020
Historique:
received:
12
06
2020
revised:
02
07
2020
accepted:
09
07
2020
entrez:
17
7
2020
pubmed:
17
7
2020
medline:
3
3
2021
Statut:
epublish
Résumé
Collagen type 1 (COL1) is a ubiquitously existing extracellular matrix protein whose high density in breast tissue favors metastasis and chemoresistance. COL1-binding of MDA-MB-231 and MCF-7 breast cancer cells is mainly dependent on β
Identifiants
pubmed: 32668815
pii: ijms21144956
doi: 10.3390/ijms21144956
pmc: PMC7404217
pii:
doi:
Substances chimiques
ABCG2 protein, human
0
ATP Binding Cassette Transporter, Subfamily G, Member 2
0
Collagen Type I
0
ITGB4 protein, human
0
Indazoles
0
Integrin beta1
0
Integrin beta4
0
Itgb1 protein, human
0
Neoplasm Proteins
0
Piperazines
0
SCH772984
0
Doxorubicin
80168379AG
Mitoxantrone
BZ114NVM5P
DDR1 protein, human
EC 2.7.10.1
Discoidin Domain Receptor 1
EC 2.7.10.1
EGFR protein, human
EC 2.7.10.1
ErbB Receptors
EC 2.7.10.1
Focal Adhesion Kinase 1
EC 2.7.10.2
PTK2 protein, human
EC 2.7.10.2
MAPK1 protein, human
EC 2.7.11.24
MAPK3 protein, human
EC 2.7.11.24
Mitogen-Activated Protein Kinase 1
EC 2.7.11.24
Mitogen-Activated Protein Kinase 3
EC 2.7.11.24
Gefitinib
S65743JHBS
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Références
Ther Adv Med Oncol. 2020 Jan 28;12:1758835919897546
pubmed: 32064003
Mol Cell. 1997 Dec;1(1):13-23
pubmed: 9659899
Cancer Cell Int. 2018 Apr 2;18:50
pubmed: 29618949
Cancer Lett. 2019 Oct 1;461:102-111
pubmed: 31319139
Nat Rev Cancer. 2020 Mar;20(3):174-186
pubmed: 31980749
Breast Cancer Res. 2014;16(5):459
pubmed: 25606594
Nat Rev Immunol. 2012 Mar 22;12(4):253-68
pubmed: 22437938
Biochim Biophys Acta Mol Cell Res. 2019 Nov;1866(11):118473
pubmed: 30954568
Oncol Lett. 2016 Nov;12(5):3598-3608
pubmed: 27900042
J Cell Physiol. 2018 Aug;233(8):6280-6290
pubmed: 29521413
Cancer Res. 2006 Aug 15;66(16):8123-30
pubmed: 16912190
Sci Rep. 2020 Feb 20;10(1):3009
pubmed: 32080212
Cell Rep. 2018 Dec 26;25(13):3674-3692.e10
pubmed: 30590041
Drug Metab Dispos. 2018 May;46(5):567-580
pubmed: 29514827
Crit Rev Oncol Hematol. 2020 Jan;145:102855
pubmed: 31927455
Sci Rep. 2017 Apr 03;7:45895
pubmed: 28368050
Cancers (Basel). 2019 Jul 12;11(7):
pubmed: 31336983
Int J Cancer. 2015 Mar 15;136(6):E508-20
pubmed: 25155634
Sci Rep. 2016 Jan 05;6:18430
pubmed: 26728650
PLoS One. 2014 Aug 29;9(8):e105792
pubmed: 25170609
Sci Rep. 2015 Nov 09;5:16408
pubmed: 26549523
Front Pharmacol. 2019 May 03;10:462
pubmed: 31130862
Histopathology. 2008 Jan;52(1):108-18
pubmed: 18171422
Am J Cancer Res. 2016 Aug 01;6(8):1609-23
pubmed: 27648353
Eur J Pharmacol. 2008 Dec 3;599(1-3):44-53
pubmed: 18938156
Respir Res. 2019 May 29;20(1):106
pubmed: 31142317
Elife. 2014 Mar 11;3:e01308
pubmed: 24618895
J Biol Chem. 2013 Mar 15;288(11):7430-7
pubmed: 23335507
EMBO J. 2003 Mar 17;22(6):1289-301
pubmed: 12628922
Fibrogenesis Tissue Repair. 2012 May 07;5(1):7
pubmed: 22564335
J Med Chem. 2013 Apr 25;56(8):3281-95
pubmed: 23521020
Cells. 2020 Feb 13;9(2):
pubmed: 32069815
BMC Cancer. 2014 Jan 02;14:1
pubmed: 24383403
Sci Rep. 2016 Nov 08;6:36336
pubmed: 27824116
Cancers (Basel). 2018 Dec 06;10(12):
pubmed: 30563275
CA Cancer J Clin. 2019 Jan;69(1):7-34
pubmed: 30620402
Invest New Drugs. 2013 Dec;31(6):1458-65
pubmed: 24068620
Cancers (Basel). 2017 Sep 16;9(9):
pubmed: 28926938
Breast Cancer Res Treat. 2015 Feb;150(1):9-18
pubmed: 25667101
BMC Cancer. 2018 Jan 6;18(1):41
pubmed: 29304770
Cell Mol Life Sci. 2011 Nov;68(22):3757-70
pubmed: 21499918
BMC Cancer. 2017 Jan 31;17(1):87
pubmed: 28143619
Ther Adv Med Oncol. 2014 Jul;6(4):154-66
pubmed: 25057302
J Invest Dermatol. 2010 Jan;130(1):74-85
pubmed: 19675578
Oncol Lett. 2018 Mar;15(3):3403-3408
pubmed: 29467865
Discov Med. 2018 May;25(139):211-223
pubmed: 29906404
Cell Adh Migr. 2018;12(4):324-334
pubmed: 29616590
Proc Natl Acad Sci U S A. 2020 Feb 18;117(7):3748-3758
pubmed: 32015106
Blood. 1999 Mar 1;93(5):1658-67
pubmed: 10029595
Eur J Med Chem. 2016 Nov 29;124:881-895
pubmed: 27676469
Exp Cell Res. 2006 Dec 10;312(20):4011-8
pubmed: 17027969
JAMA. 2019 Jan 22;321(3):288-300
pubmed: 30667505
Cell Rep. 2015 Apr 21;11(3):390-404
pubmed: 25865888
Cancer Res. 2010 Jan 15;70(2):440-6
pubmed: 20068163
Nat Rev Cancer. 2009 Sep;9(9):665-74
pubmed: 19693095
Med Oncol. 2012 Jun;29(2):401-5
pubmed: 21264531
Mol Cancer Ther. 2017 Nov;16(11):2473-2485
pubmed: 28864681
Matrix Biol. 2014 Feb;34:185-92
pubmed: 24361528
Biochim Biophys Acta Mol Cell Res. 2020 May;1867(5):118663
pubmed: 31987794
Front Pharmacol. 2016 Mar 14;7:55
pubmed: 27014069
Cancers (Basel). 2018 Nov 28;10(12):
pubmed: 30487436
Eur J Cancer. 2002 Dec;38(18):2362-70
pubmed: 12460779
PLoS One. 2012;7(12):e52209
pubmed: 23284937
Oncotarget. 2017 Jun 28;8(40):67553-67566
pubmed: 28978053
Methods Mol Biol. 2014;1204:145-53
pubmed: 25182768
Int Rev Cell Mol Biol. 2014;310:39-87
pubmed: 24725424
Mod Pathol. 2014 Sep;27(9):1212-22
pubmed: 24406864
Blood. 2013 Dec 19;122(26):4237-45
pubmed: 24136166
J Ovarian Res. 2017 Jul 25;10(1):50
pubmed: 28743276