Micro and nanoscale technologies in oral drug delivery.
Drug delivery devices
Micro and nanocarriers
Micro and nanoscale technologies
Oral drug delivery
Tissue models
Journal
Advanced drug delivery reviews
ISSN: 1872-8294
Titre abrégé: Adv Drug Deliv Rev
Pays: Netherlands
ID NLM: 8710523
Informations de publication
Date de publication:
2020
2020
Historique:
received:
23
04
2020
revised:
13
07
2020
accepted:
17
07
2020
pubmed:
25
7
2020
medline:
5
8
2021
entrez:
25
7
2020
Statut:
ppublish
Résumé
Oral administration is a pillar of the pharmaceutical industry and yet it remains challenging to administer hydrophilic therapeutics by the oral route. Smart and controlled oral drug delivery could bypass the physiological barriers that limit the oral delivery of these therapeutics. Micro- and nanoscale technologies, with an unprecedented ability to create, control, and measure micro- or nanoenvironments, have found tremendous applications in biology and medicine. In particular, significant advances have been made in using these technologies for oral drug delivery. In this review, we briefly describe biological barriers to oral drug delivery and micro and nanoscale fabrication technologies. Micro and nanoscale drug carriers fabricated using these technologies, including bioadhesives, microparticles, micropatches, and nanoparticles, are described. Other applications of micro and nanoscale technologies are discussed, including fabrication of devices and tissue engineering models to precisely control or assess oral drug delivery in vivo and in vitro, respectively. Strategies to advance translation of micro and nanotechnologies into clinical trials for oral drug delivery are mentioned. Finally, challenges and future prospects on further integration of micro and nanoscale technologies with oral drug delivery systems are highlighted.
Identifiants
pubmed: 32707147
pii: S0169-409X(20)30096-X
doi: 10.1016/j.addr.2020.07.012
pmc: PMC7374157
pii:
doi:
Substances chimiques
Drug Carriers
0
Pharmaceutical Preparations
0
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Review
Langues
eng
Sous-ensembles de citation
IM
Pagination
37-62Subventions
Organisme : Medical Research Council
ID : MR/R015651/1
Pays : United Kingdom
Organisme : British Heart Foundation
ID : RE/18/4/34215
Pays : United Kingdom
Informations de copyright
Copyright © 2020. Published by Elsevier B.V.
Références
Lab Chip. 2008 May;8(5):741-6
pubmed: 18432344
Expert Opin Biol Ther. 2004 Jan;4(1):35-51
pubmed: 14680467
J Control Release. 2017 Dec 28;268:343-351
pubmed: 29054373
Acta Pharm Sin B. 2019 Sep;9(5):902-922
pubmed: 31649842
Transplant Proc. 2011 Nov;43(9):3262-4
pubmed: 22099771
Adv Drug Deliv Rev. 2013 Jun 15;65(6):880-90
pubmed: 23220325
J Control Release. 2014 Jan 10;173:1-9
pubmed: 24096018
Proc Natl Acad Sci U S A. 2006 Feb 21;103(8):2480-7
pubmed: 16477028
Drug Discov Today. 2011 Nov;16(21-22):991-7
pubmed: 21683153
Anal Chem. 2010 Dec 15;82(24):9983-8
pubmed: 21090751
Acta Biomater. 2018 Jul 1;74:344-359
pubmed: 29723705
Adv Mater. 2016 Jun;28(21):4134-41
pubmed: 27001745
J Mater Sci Mater Med. 2008 May;19(5):2131-6
pubmed: 17999035
Biomaterials. 2012 Jun;33(19):4889-906
pubmed: 22498300
Small. 2009 Dec;5(24):2857-63
pubmed: 19787677
PDA J Pharm Sci Technol. 2012 Sep-Oct;66(5):466-500
pubmed: 23035030
J Control Release. 2006 Nov;116(1):1-27
pubmed: 17050027
J Control Release. 2000 Dec 3;69(3):445-54
pubmed: 11102684
Int J Pharm. 2013 Apr 15;447(1-2):75-93
pubmed: 23428883
Angew Chem Int Ed Engl. 2014 Jul 28;53(31):8045-8049
pubmed: 24634136
Bioorg Med Chem. 2012 Sep 15;20(18):5343-51
pubmed: 22222160
J Mater Chem B. 2013;1(14):1878-1884
pubmed: 23730504
ScientificWorldJournal. 2014 Jan 16;2014:268107
pubmed: 24550699
Biomaterials. 2012 Feb;33(5):1663-72
pubmed: 22116000
Int J Cancer. 2017 Aug 1;141(3):428-436
pubmed: 28247946
Pharmaceutics. 2018 Dec 06;10(4):
pubmed: 30563197
Int Immunopharmacol. 2008 Jun;8(6):900-8
pubmed: 18442796
J Control Release. 2000 Jan 3;63(1-2):135-40
pubmed: 10640587
Adv Drug Deliv Rev. 2018 Jul;132:139-168
pubmed: 29778901
Eur J Pharm Biopharm. 2008 Nov;70(3):777-83
pubmed: 18644444
Bioconjug Chem. 2005 Jul-Aug;16(4):1027-33
pubmed: 16029046
J Biomed Mater Res A. 2003 Nov 1;67(2):369-75
pubmed: 14619915
J Control Release. 2014 Sep 28;190:3-8
pubmed: 24794901
Acta Biomater. 2018 Jun;73:38-51
pubmed: 29653217
Adv Healthc Mater. 2018 Jan;7(2):
pubmed: 29034591
Lab Chip. 2018 Jul 10;18(14):2036-2046
pubmed: 29881844
Sci Transl Med. 2019 Nov 13;11(518):
pubmed: 31723037
J Control Release. 2019 Mar 10;297:71-78
pubmed: 30707901
J Microencapsul. 2011;28(1):62-73
pubmed: 21171817
J Control Release. 2015 Dec 10;219:431-444
pubmed: 26244713
Nat Rev Microbiol. 2007 Mar;5(3):209-18
pubmed: 17304250
Biomacromolecules. 2007 Jan;8(1):202-8
pubmed: 17206808
Expert Opin Drug Deliv. 2012 Oct;9(10):1289-304
pubmed: 22897647
Integr Biol (Camb). 2011 Dec;3(12):1224-32
pubmed: 22076329
PLoS One. 2018 May 10;13(5):e0197101
pubmed: 29746551
Biomaterials. 2008 May;29(13):1989-2006
pubmed: 18281090
Drug Dev Ind Pharm. 2002 Mar;28(3):339-44
pubmed: 12026226
J Control Release. 2005 Dec 5;109(1-3):127-38
pubmed: 16274828
Nat Med. 2019 Oct;25(10):1471-1472
pubmed: 31591600
J Control Release. 2016 Oct 10;239:27-38
pubmed: 27527555
J Control Release. 2003 Mar 7;88(2):215-28
pubmed: 12628329
Drug Discov Today. 2008 Jan;13(1-2):1-13
pubmed: 18190858
Proc Natl Acad Sci U S A. 2016 Jan 5;113(1):E7-15
pubmed: 26668389
Pharm Res. 2015 Feb;32(2):389-402
pubmed: 25082210
J Tissue Eng Regen Med. 2014 Jan;8(1):1-14
pubmed: 22711442
ACS Nano. 2012 Sep 25;6(9):7832-41
pubmed: 22900471
Am J Physiol Gastrointest Liver Physiol. 2014 Jun 1;306(11):G947-58
pubmed: 24722904
Biomaterials. 2007 Apr;28(13):2233-43
pubmed: 17261330
Eur J Pharm Sci. 2012 Sep 29;47(2):359-66
pubmed: 22771544
Biosci Trends. 2020 Mar 16;14(1):72-73
pubmed: 32074550
Sci Rep. 2019 Jul 9;9(1):9936
pubmed: 31289365
Acta Biomater. 2017 Jan 15;48:238-246
pubmed: 27815166
J Control Release. 2015 Nov 10;217:308-14
pubmed: 26390808
J Pharm Pharmacol. 2018 Feb;70(2):197-213
pubmed: 29193053
Front Bioeng Biotechnol. 2019 Jun 18;7:144
pubmed: 31275931
Eur J Pharm Biopharm. 2015 Jun;93:118-26
pubmed: 25843239
Biosens Bioelectron. 2017 Jan 15;87:865-873
pubmed: 27657849
J Control Release. 2006 Feb 21;110(3):587-94
pubmed: 16325951
Adv Drug Deliv Rev. 2009 Dec 17;61(15):1391-401
pubmed: 19758574
ACS Appl Mater Interfaces. 2013 Nov 27;5(22):12127-34
pubmed: 24175755
Chem Soc Rev. 2014 May 21;43(10):3595-629
pubmed: 24626293
Adv Drug Deliv Rev. 2012 May 1;64(6):496-507
pubmed: 22166590
Adv Drug Deliv Rev. 2016 Jun 1;101:75-88
pubmed: 27037063
Science. 2019 Oct 18;366(6463):360-364
pubmed: 31624211
ACS Nano. 2020 Feb 25;14(2):1520-1532
pubmed: 31904931
Small. 2009 Aug 3;5(15):1706-21
pubmed: 19572330
Adv Drug Deliv Rev. 2003 Feb 24;55(3):315-28
pubmed: 12628319
Int J Pharm. 2017 Jun 15;525(1):5-11
pubmed: 28377316
Bioeng Transl Med. 2016 Aug 19;1(3):338-346
pubmed: 29313019
Int J Pharm. 2014 Oct 1;473(1-2):627-35
pubmed: 25089510
J Control Release. 2004 Jul 23;98(1):37-45
pubmed: 15245887
Curr Pharm Des. 2018;24(42):5049-5061
pubmed: 30636582
J Control Release. 2016 Jan 10;221:18-25
pubmed: 26616761
Int J Food Microbiol. 2010 Jul 31;141 Suppl 1:S4-14
pubmed: 20444515
Mater Today Bio. 2019 May 25;1:100008
pubmed: 32159140
Acta Biomater. 2019 Sep 15;96:149-160
pubmed: 31252172
Pharm Dev Technol. 2000;5(1):77-85
pubmed: 10669921
ACS Appl Mater Interfaces. 2016 Jun 1;8(21):13282-93
pubmed: 27158834
Molecules. 2012 Apr 18;17(4):4612-24
pubmed: 22513487
Adv Mater. 2014 Jul 9;26(26):4497-503
pubmed: 24737409
Nanomedicine. 2014 Jan;10(1):167-76
pubmed: 23891617
Carbohydr Polym. 2016 Nov 20;153:526-534
pubmed: 27561525
Nat Commun. 2012;3:1282
pubmed: 23250412
Pharm Res. 2019 Apr 19;36(6):89
pubmed: 31004235
Polymers (Basel). 2011 Sep 1;3(3):1377-1397
pubmed: 22577513
J Pharm Sci. 1998 Aug;87(8):922-5
pubmed: 9687334
Eur J Pharm Sci. 2018 Jul 30;120:40-52
pubmed: 29678613
Eur J Pharm Biopharm. 2019 Dec;145:76-84
pubmed: 31639417
Int J Biol Macromol. 2011 Apr 1;48(3):381-5
pubmed: 20955728
Eur J Pharm Sci. 2003 Jan;18(1):89-96
pubmed: 12554077
Biotechnol J. 2011 Dec;6(12):1477-87
pubmed: 22076813
J Control Release. 2003 Apr 29;89(2):151-65
pubmed: 12711440
Assay Drug Dev Technol. 2014 May;12(4):207-18
pubmed: 24831787
Eur J Pharm Biopharm. 2012 Jun;81(2):265-72
pubmed: 22369880
J Drug Target. 2013 Aug;21(7):611-29
pubmed: 23869879
Biosens Bioelectron. 2014 Sep 15;59:166-73
pubmed: 24727602
Sci Rep. 2016 Sep 13;6:33148
pubmed: 27619235
Int J Pharm. 2001 Aug 14;224(1-2):61-7
pubmed: 11472815
Sci Rep. 2017 Oct 2;7(1):12515
pubmed: 28970586
Mol Ther Nucleic Acids. 2012 Aug 14;1:e37
pubmed: 23344179
Expert Opin Drug Deliv. 2017 Jul;14(7):851-864
pubmed: 27730820
Nat Commun. 2015 Sep 22;6:8292
pubmed: 26392213
Int J Pharm. 2008 Feb 4;348(1-2):169-74
pubmed: 17706903
Adv Drug Deliv Rev. 2013 Nov;65(11-12):1403-19
pubmed: 23726943
Int J Pharm. 2016 Sep 10;511(1):462-472
pubmed: 27418563
J Enzyme Inhib Med Chem. 2008 Oct;23(5):623-8
pubmed: 18821252
Int J Nanomedicine. 2006;1(3):297-315
pubmed: 17717971
Carbohydr Polym. 2018 Jun 15;190:240-247
pubmed: 29628244
Sci Rep. 2018 Feb 13;8(1):2871
pubmed: 29440725
Int J Pharm. 2011 May 30;410(1-2):138-44
pubmed: 21392565
Curr Opin Chem Eng. 2015 Feb;7:101-112
pubmed: 31692947
Proc SPIE Int Soc Opt Eng. 2020 Feb;11251:
pubmed: 32528214
Colloids Surf B Biointerfaces. 2019 May 1;177:284-293
pubmed: 30769230
Chemphyschem. 2009 Oct 5;10(14):2405-9
pubmed: 19705393
Int J Pharm. 2015 Oct 30;494(2):568-577
pubmed: 25498157
Pharmaceutics. 2019 Mar 19;11(3):
pubmed: 30893852
Pharm Res. 2010 Apr;27(4):576-88
pubmed: 20143253
Int Sch Res Notices. 2015 Jan 12;2015:261476
pubmed: 27347511
J Diabetes Sci Technol. 2009 Nov 01;3(6):1451-9
pubmed: 20144401
Lab Chip. 2012 Jun 21;12(12):2165-74
pubmed: 22434367
Pharmaceutics. 2019 Jul 18;11(7):
pubmed: 31323777
Pharm Res. 2006 Mar;23(3):557-64
pubmed: 16388405
Artif Cells Nanomed Biotechnol. 2016 Jun;44(4):1098-108
pubmed: 25749277
Cell Stem Cell. 2018 Mar 1;22(3):310-324
pubmed: 29499151
Nat Med. 2019 Oct;25(10):1512-1518
pubmed: 31591601
J Control Release. 2004 May 31;97(1):115-24
pubmed: 15147809
Adv Drug Deliv Rev. 2005 Nov 3;57(11):1583-94
pubmed: 16169120
Int J Pharm. 1999 Jul 5;184(1):73-84
pubmed: 10425353
Adv Drug Deliv Rev. 2012 May 1;64(6):557-70
pubmed: 22212900
J Pharm Sci. 2019 Sep;108(9):3138-3145
pubmed: 31034907
Curr Opin Pharmacol. 2017 Oct;36:58-65
pubmed: 28850875
Mater Sci Eng C Mater Biol Appl. 2017 Sep 1;78:420-428
pubmed: 28576004
Nat Rev Drug Discov. 2002 Jan;1(1):77-84
pubmed: 12119612
Biomed Microdevices. 2017 Jun;19(2):37
pubmed: 28451924
Nat Biomed Eng. 2020 Jan;4(1):84-96
pubmed: 31686002
J Pharm Sci. 2016 Jul;105(7):2155-63
pubmed: 27290630
Eur J Pharm Sci. 2005 Jul-Aug;25(4-5):445-53
pubmed: 15890503
ACS Nano. 2016 Jun 28;10(6):5873-81
pubmed: 27268699
Int J Nanomedicine. 2012;7:1851-63
pubmed: 22605934
Science. 2019 Feb 8;363(6427):611-615
pubmed: 30733413
J Pharm (Cairo). 2014;2014:904036
pubmed: 26556206
Adv Drug Deliv Rev. 2018 Mar 15;128:3-28
pubmed: 28919029
Nano Lett. 2013 Jan 9;13(1):164-71
pubmed: 23186530
Toxicol In Vitro. 2014 Aug;28(5):885-95
pubmed: 24662032
Adv Mater. 2020 Apr;32(13):e1901935
pubmed: 31222910
Pharm Sci Technol Today. 2000 Apr;3(4):138-145
pubmed: 10754543
Nat Rev Drug Discov. 2006 Mar;5(3):210-8
pubmed: 16518374
J Mech Behav Biomed Mater. 2018 Aug;84:74-87
pubmed: 29751274
Carbohydr Polym. 2017 Aug 1;169:157-166
pubmed: 28504131
Biomacromolecules. 2007 Sep;8(9):2845-50
pubmed: 17665945
Nat Biotechnol. 2014 Aug;32(8):760-72
pubmed: 25093883
Acta Biomater. 2014 Mar;10(3):1324-32
pubmed: 24287161
Anal Sci. 2009 Dec;25(12):1403-7
pubmed: 20009325
J Pharmacol Exp Ther. 2019 Sep;370(3):529-543
pubmed: 31010845
J Control Release. 2017 Dec 28;268:10-18
pubmed: 29030223
Eur J Pharm Biopharm. 2007 Mar;65(3):379-87
pubmed: 17123802
Eur J Pharm Sci. 2017 Sep 30;107:148-167
pubmed: 28690099
Lab Chip. 2014 Jul 7;14(13):2145-60
pubmed: 24647678
Int J Pharm. 2007 Apr 20;335(1-2):167-175
pubmed: 17161566
Micromachines (Basel). 2019 Oct 09;10(10):
pubmed: 31601016
Eur J Pharm Biopharm. 2007 Jan;65(1):10-7
pubmed: 17101268
Drug Dev Ind Pharm. 2016;42(7):1019-31
pubmed: 26625986
Micromachines (Basel). 2019 Sep 10;10(9):
pubmed: 31510012
Eur J Pharm Biopharm. 2011 Sep;79(1):197-204
pubmed: 21345371
ACS Nano. 2019 Feb 26;13(2):1324-1332
pubmed: 30689352
Drug Deliv. 2016 Sep;23(7):2541-2554
pubmed: 25853478
ACS Biomater Sci Eng. 2017 Sep 11;3(9):2144-2154
pubmed: 33440563
Nat Commun. 2017 Aug 16;8(1):272
pubmed: 28814725
J Pharm Sci. 2003 Aug;92(8):1614-23
pubmed: 12884248
Int J Pharm. 2015 Oct 30;494(2):611-618
pubmed: 25526674
Lab Chip. 2010 Apr 21;10(8):939-56
pubmed: 20358102
Daru. 2011;19(6):385-403
pubmed: 23008684
Drug Des Devel Ther. 2015 Feb 10;9:791-8
pubmed: 25709403
Biomaterials. 2008 Feb;29(4):475-86
pubmed: 17953985
Eur J Pharm Biopharm. 2017 May;114:135-144
pubmed: 28111241
Colloids Surf B Biointerfaces. 2013 Jan 1;101:353-60
pubmed: 23010041
Biomaterials. 2018 Sep;178:134-146
pubmed: 29929183
J Drug Target. 2009 Apr;17(3):249-56
pubmed: 19255893
Adv Drug Deliv Rev. 2001 Apr 25;47(2-3):165-96
pubmed: 11311991
Phytomedicine. 2014 Oct 15;21(12):1627-32
pubmed: 25442269
Acta Biomater. 2008 Sep;4(5):1126-38
pubmed: 18474452
J Cell Physiol. 1996 Aug;168(2):476-88
pubmed: 8707883
Adv Drug Deliv Rev. 2004 Sep 22;56(11):1621-33
pubmed: 15350292
J Pharm Sci. 2015 Feb;104(2):362-7
pubmed: 25250829
J Control Release. 2006 Mar 10;111(1-2):41-6
pubmed: 16377016
Int J Pharm. 2009 Mar 18;369(1-2):53-63
pubmed: 19084583
Acta Biomater. 2009 Mar;5(3):817-31
pubmed: 19010748
ACS Biomater Sci Eng. 2020 Apr 13;6(4):2478-2486
pubmed: 33455326
Diabetes Obes Metab. 2000 Aug;2(4):243-50
pubmed: 11225658
Acta Biomater. 2010 Aug;6(8):3072-80
pubmed: 20144748
Adv Drug Deliv Rev. 2001 Dec 3;53(1):95-108
pubmed: 11733119
Int J Pharm. 2005 Apr 27;294(1-2):247-59
pubmed: 15814248
Nat Commun. 2018 Jan 9;9(1):2
pubmed: 29317618
Trends Biotechnol. 2014 Jan;32(1):32-45
pubmed: 24210498
Small. 2007 Mar;3(3):412-8
pubmed: 17285662
Pharm Res. 2008 Oct;25(10):2370-8
pubmed: 18663411
J Control Release. 2008 Jul 2;129(1):1-10
pubmed: 18499294
Mol Pharm. 2015 Nov 2;12(11):4077-84
pubmed: 26473653
J Pharm Sci. 2019 Jul;108(7):2238-2242
pubmed: 30779888
Mol Pharm. 2010 Jun 7;7(3):642-51
pubmed: 20205474
Int J Nanomedicine. 2019 Sep 04;14:7191-7213
pubmed: 31564873
Wiley Interdiscip Rev Nanomed Nanobiotechnol. 2017 Jan;9(1):
pubmed: 27312983
Eur J Pharm Biopharm. 2012 Jan;80(1):95-102
pubmed: 21964316
J Control Release. 2004 Mar 24;95(3):447-53
pubmed: 15023456
Cancer Res Treat. 2014 Jan;46(1):2-18
pubmed: 24520218
Adv Drug Deliv Rev. 2013 Nov;65(11-12):1575-88
pubmed: 23856409
Biomaterials. 2001 Apr;22(7):687-94
pubmed: 11246962
Int J Pharm. 2015 Jul 25;490(1-2):384-90
pubmed: 26043827
N Engl J Med. 2020 Jun 11;382(24):2327-2336
pubmed: 32275812
J Drug Target. 2013 Jul;21(6):515-27
pubmed: 23621127
Front Pharmacol. 2017 May 23;8:287
pubmed: 28588490
J Microencapsul. 2012;29(2):147-55
pubmed: 22126315
Clin Pharmacokinet. 2001;40(2):77-84
pubmed: 11286325
ACS Nano. 2015 Aug 25;9(8):8291-302
pubmed: 26235314
Int J Pharm. 2015 Jul 15;489(1-2):277-84
pubmed: 25957702
Pharm Res. 2007 Jan;24(1):1-16
pubmed: 17109211
Adv Healthc Mater. 2018 Sep;7(17):e1800285
pubmed: 29984479
J Control Release. 2012 Nov 10;163(3):361-7
pubmed: 23041274
Front Pharmacol. 2016 Jun 28;7:185
pubmed: 27445821
Adv Drug Deliv Rev. 2011 Apr 30;63(4-5):352-66
pubmed: 21241756
Proc Natl Acad Sci U S A. 2003 Sep 16;100(19):10603-6
pubmed: 12960386
P T. 2017 Dec;42(12):742-755
pubmed: 29234213
Int J Nanomedicine. 2011;6:1155-66
pubmed: 21822379
Diabetes Care. 2010 Feb;33(2):240-5
pubmed: 20103556
Int J Antimicrob Agents. 2020 Jul;56(1):105949
pubmed: 32205204
Biomed Microdevices. 2015;17(3):9958
pubmed: 25981751