Effects of Standardized Medicinal Plant Extracts on Drug Metabolism Mediated by CYP3A4 and CYP2D6 Enzymes.


Journal

Chemical research in toxicology
ISSN: 1520-5010
Titre abrégé: Chem Res Toxicol
Pays: United States
ID NLM: 8807448

Informations de publication

Date de publication:
21 09 2020
Historique:
pubmed: 14 8 2020
medline: 24 8 2021
entrez: 14 8 2020
Statut: ppublish

Résumé

The use of medicinal plants concomitantly with conventional drugs can result in herb-drug interactions that cause fluctuations in drug bioavailability and consequent therapeutic failure and/or toxic effects. The CYP superfamily of enzymes plays an important role in herb-drug interactions. Among CYP enzymes, CYP3A4 and CYP2D6 are the most relevant since they metabolize about 50% and 30% of the drugs on the market, respectively. Thus, the main goal of this study was to evaluate the occurrence of

Identifiants

pubmed: 32786546
doi: 10.1021/acs.chemrestox.0c00182
doi:

Substances chimiques

Cytochrome P-450 Enzyme Inhibitors 0
Plant Extracts 0
Recombinant Proteins 0
Cytochrome P-450 CYP2D6 EC 1.14.14.1
Cytochrome P-450 CYP3A EC 1.14.14.1

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

2408-2419

Auteurs

Clarissa Feltrin (C)

Programa de Pós-Graduação em Farmácia, Centro de Ciências da Saúde, Universidade Federal de Santa Catarina, Florianópolis, 88040-900, Santa Catarina, Brazil.

Ingrid Vicente Farias (IV)

Programa de Pós-Graduação em Farmácia, Centro de Ciências da Saúde, Universidade Federal de Santa Catarina, Florianópolis, 88040-900, Santa Catarina, Brazil.

Louis Pergaud Sandjo (LP)

Departamento de Química, Universidade Federal de Santa Catarina, Florianópolis, 88040-900, Santa Catarina, Brazil.

Flávio Henrique Reginatto (FH)

Programa de Pós-Graduação em Farmácia, Centro de Ciências da Saúde, Universidade Federal de Santa Catarina, Florianópolis, 88040-900, Santa Catarina, Brazil.

Cláudia Maria Oliveira Simões (CMO)

Programa de Pós-Graduação em Farmácia, Centro de Ciências da Saúde, Universidade Federal de Santa Catarina, Florianópolis, 88040-900, Santa Catarina, Brazil.

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Classifications MeSH