The African natural product knipholone anthrone and its analogue anthralin (dithranol) enhance HIV-1 latency reversal.
drug discovery
drug-drug synergy
histone deacetylase (HDAC)
histone deacetylase inhibitor (HDAC inhibitor) (HDI)
human immunodeficiency virus (HIV)
latency reversal
molecular pharmacology
natural product
protein kinase C (PKC)
viral reservoirs
Journal
The Journal of biological chemistry
ISSN: 1083-351X
Titre abrégé: J Biol Chem
Pays: United States
ID NLM: 2985121R
Informations de publication
Date de publication:
09 10 2020
09 10 2020
Historique:
received:
12
02
2020
revised:
06
08
2020
pubmed:
14
8
2020
medline:
17
2
2021
entrez:
14
8
2020
Statut:
ppublish
Résumé
A sterilizing or functional cure for HIV is currently precluded by resting CD4
Identifiants
pubmed: 32788215
pii: S0021-9258(17)49805-X
doi: 10.1074/jbc.RA120.013031
pmc: PMC7549037
doi:
Substances chimiques
Anthracenes
0
knipholone anthrone
0
Anthralin
U8CJK0JH5M
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
14084-14099Subventions
Organisme : NIAID NIH HHS
ID : UM1 AI126620
Pays : United States
Organisme : NINDS NIH HHS
ID : R21 NS106970
Pays : United States
Organisme : NIA NIH HHS
ID : R01 AG062383
Pays : United States
Organisme : NIDDK NIH HHS
ID : R01 DK123733
Pays : United States
Organisme : NIAID NIH HHS
ID : R21 AI143385
Pays : United States
Organisme : NIAID NIH HHS
ID : P30 AI045008
Pays : United States
Organisme : NIAID NIH HHS
ID : R21 AI129636
Pays : United States
Organisme : NINDS NIH HHS
ID : R01 NS117458
Pays : United States
Organisme : Wellcome Trust
Pays : United Kingdom
Organisme : CIHR
ID : PJT-153057
Pays : Canada
Organisme : CIHR
ID : PJT-159625
Pays : Canada
Organisme : Wellcome Trust
ID : 107752/Z/15/Z
Pays : United Kingdom
Informations de copyright
© 2020 Richard et al.
Déclaration de conflit d'intérêts
Conflict of interest—The authors declare that they have no conflicts of interest with the contents of this article.
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