Photoswitchable Lipids.

amphiphiles azobenzene lipids photopharmacology photoswitches

Journal

Chembiochem : a European journal of chemical biology
ISSN: 1439-7633
Titre abrégé: Chembiochem
Pays: Germany
ID NLM: 100937360

Informations de publication

Date de publication:
05 01 2021
Historique:
received: 08 07 2020
revised: 11 08 2020
pubmed: 14 8 2020
medline: 24 9 2021
entrez: 14 8 2020
Statut: ppublish

Résumé

Photoswitchable lipids are emerging tools for the precise manipulation and study of lipid function. They can modulate many aspects of membrane biophysics, including permeability, fluidity, lipid mobility and domain formation. They are also very useful in lipid physiology and enable optical control of a wide array of lipid receptors, such as ion channels, G protein-coupled receptors, nuclear hormone receptors, and enzymes that translocate to membranes. Enzymes involved in lipid metabolism often process them in a light-dependent fashion. Photoswitchable lipids complement other functionalized lipids widely used in lipid chemical biology, including isotope-labeled lipids (lipidomics), fluorescent lipids (imaging), bifunctional lipids (lipid-protein crosslinking), photocaged lipids (photopharmacology), and other labeled variants.

Identifiants

pubmed: 32790211
doi: 10.1002/cbic.202000449
doi:

Substances chimiques

Lipids 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't Review

Langues

eng

Sous-ensembles de citation

IM

Pagination

73-83

Informations de copyright

© 2020 Wiley-VCH GmbH.

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Auteurs

Johannes Morstein (J)

Department of Chemistry, New York University, 100 Washington Square East, New York, NY, 10003-6699, USA.

Anna C Impastato (AC)

Department of Chemistry, New York University, 100 Washington Square East, New York, NY, 10003-6699, USA.

Dirk Trauner (D)

Department of Chemistry, New York University, 100 Washington Square East, New York, NY, 10003-6699, USA.

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Classifications MeSH