Synthesis, docking study and biological evaluation of ᴅ-fructofuranosyl and ᴅ-tagatofuranosyl sulfones as potential inhibitors of the mycobacterial galactan synthesis targeting the galactofuranosyltransferase GlfT2.
GlfT2
molecular modeling
mycobacterium tuberculosis
synthesis
transition state inhibitors
Journal
Beilstein journal of organic chemistry
ISSN: 1860-5397
Titre abrégé: Beilstein J Org Chem
Pays: Germany
ID NLM: 101250746
Informations de publication
Date de publication:
2020
2020
Historique:
received:
30
04
2020
accepted:
09
07
2020
entrez:
18
8
2020
pubmed:
18
8
2020
medline:
18
8
2020
Statut:
epublish
Résumé
A series of ten novel ᴅ-fructofuranosyl and ᴅ-tagatofuranosyl sulfones bearing a 1-
Identifiants
pubmed: 32802202
doi: 10.3762/bjoc.16.152
pmc: PMC7404141
doi:
Types de publication
Journal Article
Langues
eng
Pagination
1853-1862Informations de copyright
Copyright © 2020, Baráth et al.; licensee Beilstein-Institut.
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