Renin-Angiotensin System and Coronavirus Disease 2019: A Narrative Review.

COVID-19 RAS inhibitors SARS-COV-2 heart damage pulmonary damage renin-angiotensin system

Journal

Frontiers in cardiovascular medicine
ISSN: 2297-055X
Titre abrégé: Front Cardiovasc Med
Pays: Switzerland
ID NLM: 101653388

Informations de publication

Date de publication:
2020
Historique:
received: 05 05 2020
accepted: 06 07 2020
entrez: 28 8 2020
pubmed: 28 8 2020
medline: 28 8 2020
Statut: epublish

Résumé

Although clinical manifestations of the 2019 novel coronavirus disease pandemic (COVID-19), caused by the novel severe acute respiratory syndrome coronavirus 2 (SARS-COV-2), are mainly respiratory symptoms, patients can also develop severe cardiovascular damage. Therefore, understanding the damage caused by SARS-COV-2 to the cardiovascular system and the underlying mechanisms is fundamental. The cardiovascular damage may be related to the imbalance of the renin-angiotensin-system (RAS) as this virus binds the Angiotensin-Converting-Enzyme 2 (ACE2), expressed on the lung alveolar epithelial cells, to enter into cells. Virus internalization may cause a downregulation of ACE2 on host cell surface that could lead to a local increased level of angiotensin II (AII) and a reduced level of angiotensin 1-7 (A1-7). An imbalance between these angiotensins may be responsible for the lung and heart damage. Pharmacological strategies that interfere with the viral attachment to ACE2 (umifenovir and hydroxychloroquine/chloroquine) or that modulate the RAS (analogous of A1-7 and ACE2, losartan) are in clinical development for COVID-19. The use of RAS inhibitors has also become a matter of public concern as these drugs may increase the mRNA expression and levels of ACE2 and impact the virulence and transmission of SARS-COV-2. Data on the effect of RAS inhibitors on ACE2 mRNA expression are scarce. Scientific societies expressed their opinion on continuing the therapy with RAS inhibitors in patients with COVID-19 and underlying cardiovascular diseases. In conclusion, RAS may play a role in SARS-COV-2-induced cardiac and pulmonary damage. Further studies are needed to better understand the role of RAS in COVID-19 and to guide decision on the use of RAS inhibitors.

Identifiants

pubmed: 32850989
doi: 10.3389/fcvm.2020.00143
pmc: PMC7431661
doi:

Types de publication

Journal Article Review

Langues

eng

Pagination

143

Informations de copyright

Copyright © 2020 Mascolo, Scavone, Rafaniello, Ferrajolo, Racagni, Berrino, Paolisso, Rossi and Capuano.

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Auteurs

Annamaria Mascolo (A)

Section of Pharmacology "L. Donatelli", Department of Experimental Medicine, University of Campania "Luigi Vanvitelli", Naples, Italy.
Campania Regional Centre for Pharmacovigilance and Pharmacoepidemiology, Naples, Italy.

Cristina Scavone (C)

Section of Pharmacology "L. Donatelli", Department of Experimental Medicine, University of Campania "Luigi Vanvitelli", Naples, Italy.
Campania Regional Centre for Pharmacovigilance and Pharmacoepidemiology, Naples, Italy.

Concetta Rafaniello (C)

Section of Pharmacology "L. Donatelli", Department of Experimental Medicine, University of Campania "Luigi Vanvitelli", Naples, Italy.
Campania Regional Centre for Pharmacovigilance and Pharmacoepidemiology, Naples, Italy.

Carmen Ferrajolo (C)

Section of Pharmacology "L. Donatelli", Department of Experimental Medicine, University of Campania "Luigi Vanvitelli", Naples, Italy.
Campania Regional Centre for Pharmacovigilance and Pharmacoepidemiology, Naples, Italy.

Giorgio Racagni (G)

Department of Pharmacological and Biomolecular Sciences, Università degli Studi di Milano, Milan, Italy.

Liberato Berrino (L)

Section of Pharmacology "L. Donatelli", Department of Experimental Medicine, University of Campania "Luigi Vanvitelli", Naples, Italy.

Giuseppe Paolisso (G)

Department of Advanced Medical and Surgical Sciences, University of Campania "Luigi Vanvitelli", Naples, Italy.

Francesco Rossi (F)

Section of Pharmacology "L. Donatelli", Department of Experimental Medicine, University of Campania "Luigi Vanvitelli", Naples, Italy.
Campania Regional Centre for Pharmacovigilance and Pharmacoepidemiology, Naples, Italy.

Annalisa Capuano (A)

Section of Pharmacology "L. Donatelli", Department of Experimental Medicine, University of Campania "Luigi Vanvitelli", Naples, Italy.
Campania Regional Centre for Pharmacovigilance and Pharmacoepidemiology, Naples, Italy.

Classifications MeSH