Sirtuin inhibition and anti-cancer activities of ethyl 2-benzimidazole-5-carboxylate derivatives.
Journal
MedChemComm
ISSN: 2040-2503
Titre abrégé: Medchemcomm
Pays: England
ID NLM: 101531525
Informations de publication
Date de publication:
01 Dec 2019
01 Dec 2019
Historique:
received:
08
06
2019
accepted:
28
10
2019
entrez:
9
9
2020
pubmed:
10
9
2020
medline:
10
9
2020
Statut:
epublish
Résumé
New benzimidazoles were synthesized based on the previously identified sirtuin inhibitor BZD9L1. The compounds were screened for their sirtuin (SIRT1, SIRT2 and SIRT3) inhibitory activities. Compound
Identifiants
pubmed: 32904142
doi: 10.1039/c9md00323a
pii: c9md00323a
pmc: PMC7451065
doi:
Types de publication
Journal Article
Langues
eng
Pagination
2140-2145Informations de copyright
This journal is © The Royal Society of Chemistry 2019.
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